SCHEMBL16622216

SCHEMBL16622216

CC(=O)Nc1cccc(C#Cc2ccc(CC(N)=O)cc2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.52
ALDH1A1 P00352 4/20 0.50
RAB9A P51151 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
GRM5 P41594 1/20 0.50
KDM4E B2RXH2 1/20 0.50
MEN1 O00255 1/20 0.50
HPGD P15428 1/20 0.50
CYP2C19 P33261 1/20 0.50
KMT2A Q03164 1/20 0.50
NLRP3 Q96P20 2/20 0.49
PTPN11 Q06124 1/20 0.49
ACACB O00763 2/20 0.47
AOC3 Q16853 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
POLB P06746 1/20 0.44
NR4A1 P22736 1/20 0.44
CYP1A2 P05177 1/20 0.44
FFAR1 O14842 1/20 0.44
HSD17B10 Q99714 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1432559 0.87 NLRP3 (0.53) IKBKBALDH1A1RAB9ASMN1; SMN2GRM5
Hydrochloric Acid SCHEMBL1432557 0.86 NLRP3 (0.52) IKBKBALDH1A1RAB9ASMN1; SMN2GRM5
SCHEMBL16622212 0.86 KMT2A (0.69) ALDH1A1RAB9ASMN1; SMN2KDM4EMEN1
SCHEMBL15612045 0.81 PTPN11 (0.71) IKBKBALDH1A1RAB9ASMN1; SMN2GRM5
SCHEMBL16622211 0.81 KDM4E (0.45) ALDH1A1RAB9ASMN1; SMN2KDM4EMEN1
SCHEMBL18130126 0.80 ALDH1A1 (0.60) IKBKBALDH1A1RAB9ASMN1; SMN2GRM5
SCHEMBL27829449 0.80 PTPN1 (0.50) IKBKBALDH1A1RAB9ASMN1; SMN2GRM5
SCHEMBL5037396 0.80 ALDH1A1 (0.57) ALDH1A1RAB9AMEN1KMT2ANLRP3
Hydrochloric Acid SCHEMBL28790880 0.79 PTPN1 (0.49) IKBKBALDH1A1RAB9ASMN1; SMN2GRM5
SCHEMBL21715154 0.77 GRM5 (0.58) IKBKBALDH1A1RAB9ASMN1; SMN2GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8999989-B2 Benzene or thiophene derivative and use thereof as VAP-1 inhibitor R-TECH UENO, LTD. (JP) 2015-04-07 US disclosed