SCHEMBL16622211

SCHEMBL16622211

CC(=O)Nc1ccc(C#Cc2ccc(CC(N)=O)cc2)cc1NC(C)=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.45
MEN1 O00255 1/20 0.45
ALDH1A1 P00352 1/20 0.45
HPGD P15428 1/20 0.45
CYP2C19 P33261 1/20 0.45
RAB9A P51151 1/20 0.45
KMT2A Q03164 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
ACACB O00763 5/20 0.41
CA2 P00918 1/20 0.40
FFAR1 O14842 1/20 0.40
NEU3 Q9UQ49 1/20 0.38
LMNA P02545 2/20 0.38
TDP1 Q9NUW8 2/20 0.38
ADRB2 P07550 1/20 0.38
ADRB1 P08588 1/20 0.38
CNR1 P21554 1/20 0.38
ADRA1D P25100 1/20 0.38
ADRA1A P35348 1/20 0.38
ADRA1B P35368 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1432853 0.86 SMN1; SMN2 (0.43) KDM4EMEN1ALDH1A1HPGDCYP2C19
Hydrochloric Acid SCHEMBL1432374 0.85 SMN1; SMN2 (0.42) KDM4EMEN1ALDH1A1HPGDCYP2C19
SCHEMBL16622212 0.82 KMT2A (0.69) KDM4EMEN1ALDH1A1HPGDCYP2C19
SCHEMBL16622220 0.82 EGLN1 (0.41) KDM4EMEN1ALDH1A1HPGDCYP2C19
SCHEMBL16622216 0.81 IKBKB (0.52) KDM4EMEN1ALDH1A1HPGDCYP2C19
SCHEMBL27829393 0.79 PTPN1 (0.43) KDM4EMEN1ALDH1A1HPGDCYP2C19
Hydrochloric Acid SCHEMBL27829445 0.78 PTPN1 (0.42) KDM4EMEN1ALDH1A1HPGDCYP2C19
SCHEMBL16622225 0.76 PTK2 (0.46) KDM4EMEN1ALDH1A1HPGDCYP2C19
SCHEMBL16622218 0.73 ACACB (0.43) KDM4EMEN1ALDH1A1HPGDCYP2C19
SCHEMBL4086221 0.72 TDP1 (0.59) KDM4EMEN1ALDH1A1HPGDCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8999989-B2 Benzene or thiophene derivative and use thereof as VAP-1 inhibitor R-TECH UENO, LTD. (JP) 2015-04-07 US disclosed