SCHEMBL16623135

SCHEMBL16623135

CC(C)(C)OC(=O)NOCc1cccc(-c2ccc(C(=O)O)cc2)c1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BCL2 P10415 3/20 0.54
AOC3 Q16853 2/20 0.51
RXRA P19793 4/20 0.48
RXRB P28702 4/20 0.48
MRGPRX4 Q96LA9 3/20 0.47
CTSB P07858 1/20 0.47
CTSS P25774 1/20 0.47
CTSK P43235 1/20 0.47
NR4A2 P43354 1/20 0.46
HDAC1 Q13547 1/20 0.45
NR1H4 Q96RI1 1/20 0.43
CYP17A1 P05093 1/20 0.43
ADRB3 P13945 1/20 0.42
GPR183 P32249 1/20 0.42
GRM2 Q14416 1/20 0.42
RXRG P48443 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4399149 0.87 MRGPRX4 (0.50) MRGPRX4NR1H4
SCHEMBL5549803 0.83 HDAC1 (0.60) BCL2AOC3RXRARXRBCTSB
SCHEMBL32665365 0.79 NQO2 (0.44)
SCHEMBL716007 0.79 NPC1 (0.56) CTSBCTSSCTSK
SCHEMBL4391966 0.79 LOXL2 (0.58) MRGPRX4
SCHEMBL19639269 0.78 CTSS (0.47) AOC3CTSBCTSSCTSKNR4A2
SCHEMBL11892918 0.78 HDAC1 (0.53) BCL2AOC3RXRARXRBCTSB
SCHEMBL19658012 0.77 CTSS (0.46) AOC3RXRACTSBCTSSCTSK
SCHEMBL17894367 0.76 CTSS (0.41) RXRARXRBMRGPRX4CTSBCTSS
SCHEMBL17894365 0.76 CTSS (0.41) RXRARXRBMRGPRX4CTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2665744-B1 MACROCYCLIC COMPOUNDS WITH A HYBRID PEPTIDIC/NON-PEPTIDIC BACKBONE AND METHODS FOR THEIR PREPARATION UNIV ROCHESTER (US) 2015-04-08 EP disclosed