SCHEMBL16623541

SCHEMBL16623541

N=C(c1csc(C(N)=O)c1)c1c(NCc2ccc(O)cc2)cc[nH]c1=O

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.34
AURKA O14965 1/20 0.31
RPS6KB1 P23443 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
THRB P10828 1/20 0.31
ALOX12 P18054 1/20 0.31
KMT2A Q03164 1/20 0.31
HPGD P15428 1/20 0.31
HTT P42858 1/20 0.31
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16623481 0.91 EGFR (0.38) EGFRKDM4EMEN1ALDH1A1MAPT
SCHEMBL16726667 0.81 HPGD (0.31) MEN1KMT2AHPGDHTT
SCHEMBL16726671 0.78 HPGD (0.34) HPGDHTT
SCHEMBL16623535 0.77 ALDH1A1 (0.36) EGFRKDM4EMEN1ALDH1A1MAPT
SCHEMBL16623523 0.76 HPGD (0.33) EGFRHPGDHTT
SCHEMBL16623551 0.76 JAK1 (0.34) CA1CA2
SCHEMBL16623467 0.76 HPGD (0.32) HPGDHTT
SCHEMBL16726703 0.76 HPGD (0.32) HPGDHTT
SCHEMBL16623575 0.76 HPGD (0.32) HPGDHTT
SCHEMBL16623536 0.75 HSP90AA1 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed
EP-2857400-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2015-04-08 EP disclosed