SCHEMBL16624030

SCHEMBL16624030

COc1ccc2c(c1)CN(C(C)C)CC2O

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 9/20 0.48
SLC6A2 P23975 6/20 0.48
SLC6A3 Q01959 6/20 0.48
HRH3 Q9Y5N1 3/20 0.45
GRIN2B Q13224 2/20 0.44
GRIN1 Q05586 1/20 0.44
KIF11 P52732 1/20 0.44
KDM2B Q8NHM5 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16624024 0.89 SLC6A4 (0.48) SLC6A4SLC6A2SLC6A3HRH3KDM2B
SCHEMBL18034964 0.82 SLC6A4 (0.63) SLC6A4SLC6A2SLC6A3HRH3GRIN2B
SCHEMBL18033538 0.81 SLC6A2 (0.47) SLC6A4SLC6A2SLC6A3KIF11
SCHEMBL18253962 0.79 CHRNB2 (0.37) SLC6A4SLC6A2SLC6A3HRH3KIF11
SCHEMBL16624052 0.78 MTNR1B (0.46) HRH3GRIN2BGRIN1KDM2B
SCHEMBL11794884 0.77 SLC6A4 (0.51) SLC6A4SLC6A2SLC6A3HRH3KIF11
Hydrochloric Acid SCHEMBL11794735 0.76 SLC6A4 (0.50) SLC6A4SLC6A2SLC6A3HRH3KIF11
SCHEMBL18252814 0.76 KCNH2 (0.43) KIF11
SCHEMBL18252817 0.76 KCNH2 (0.43) KIF11
SCHEMBL18252841 0.76 KCNH2 (0.43) KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3053917-A1 T-TYPE CALCIUM CHANNEL BLOCKER Nissan Chemical Industries, Ltd. (JP) 2016-08-10 EP disclosed
WO-2015050212-A1 T-TYPE CALCIUM CHANNEL BLOCKER 日産化学工業株式会社 2015-04-09 WO disclosed