SCHEMBL16624873

SCHEMBL16624873

C[C@]1(COc2ccc(-n3cc(-c4ccccc4)nn3)cc2)Cn2cc(I)nc2O1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.42
PTGS2 P35354 4/20 0.40
PTGS1 P23219 3/20 0.40
TSHR P16473 2/20 0.39
LMNA P02545 1/20 0.39
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
CA1 P00915 3/20 0.38
CA2 P00918 3/20 0.38
CA9 Q16790 2/20 0.38
CA5A P35218 2/20 0.38
CA5B Q9Y2D0 2/20 0.38
CA12 O43570 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
OGT O15294 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16624950 0.93 KCNH2 (0.42) KCNH2PTGS2PTGS1SLC6A2SLC6A4
SCHEMBL16624945 0.89 FLT3 (0.49) KCNH2PTGS2PTGS1SLC6A2SLC6A4
SCHEMBL16624985 0.89 KCNH2 (0.56) KCNH2PTGS2PTGS1SLC6A2SLC6A4
SCHEMBL16624874 0.87 KCNH2 (0.43) KCNH2PTGS1SLC6A2SLC6A4CA1
SCHEMBL18031081 0.85 KCNH2 (0.63) KCNH2PTGS2PTGS1SLC6A2SLC6A4
SCHEMBL16618280 0.78 KCNH2 (0.63) KCNH2PTGS2PTGS1SLC6A2SLC6A4
SCHEMBL16618251 0.77 KCNH2 (0.62) KCNH2PTGS2PTGS1SLC6A2SLC6A4
SCHEMBL16624949 0.77 KCNH2 (0.63) KCNH2PTGS2PTGS1SLC6A2SLC6A4
SCHEMBL18011988 0.76 KCNH2 (0.62) KCNH2PTGS2PTGS1SLC6A2SLC6A4
SCHEMBL16618234 0.76 KCNH2 (0.60) KCNH2PTGS1SLC6A2SLC6A4CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015049693-A1 6-NITRO-2,3-DIHYDROIMIDAZO[2,1-b]OXAZOLES AND A PROCESS FOR THE PREPARATION THEREOF COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2015-04-09 WO disclosed