SCHEMBL16624874

SCHEMBL16624874

C[C@]1(COc2ccc(-n3cc(-c4cccc(C(F)(F)F)c4)nn3)cc2)Cn2cc(I)nc2O1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42
KEAP1 Q14145 1/20 0.41
NFE2L2 Q16236 1/20 0.41
PTGS1 P23219 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
GPR55 Q9Y2T6 1/20 0.39
KDR P35968 1/20 0.37
TEK Q02763 1/20 0.37
AURKA O14965 5/20 0.37
AURKB Q96GD4 3/20 0.37
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC8 Q9BY41 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16624873 0.87 KCNH2 (0.42) KCNH2CA12CA1CA2CA9
SCHEMBL18011979 0.87 KCNH2 (0.62) KCNH2CA12CA1CA2CA9
SCHEMBL16624985 0.85 KCNH2 (0.56) KCNH2CA12CA1CA2CA9
SCHEMBL16624950 0.84 KCNH2 (0.42) KCNH2CA12CA1CA2CA9
SCHEMBL16624945 0.81 FLT3 (0.49) KCNH2PTGS1SLC6A2SLC6A4RXRA
SCHEMBL18031082 0.77 KCNH2 (0.70) KCNH2KEAP1NFE2L2PTGS1SLC6A2
SCHEMBL16618234 0.77 KCNH2 (0.60) KCNH2CA12CA9KEAP1NFE2L2
SCHEMBL16618336 0.74 KCNH2 (0.58) KCNH2CA12CA9KEAP1NFE2L2
SCHEMBL18031081 0.74 KCNH2 (0.63) KCNH2CA12CA1CA2CA9
SCHEMBL16618270 0.72 KCNH2 (0.78) KCNH2CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015049693-A1 6-NITRO-2,3-DIHYDROIMIDAZO[2,1-b]OXAZOLES AND A PROCESS FOR THE PREPARATION THEREOF COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2015-04-09 WO disclosed