SCHEMBL16625694

SCHEMBL16625694

Brc1ccc2c(c1)C1(c3cc(Br)ccc3-2)c2cc(Br)ccc2-c2ccc(I)cc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.40
S100A4 P26447 1/20 0.35
AKR1A1 P14550 1/20 0.35
AKR1B1 P15121 1/20 0.35
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA4 P22748 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
TDP2 O95551 3/20 0.34
CCNB2 O95067 1/20 0.32
CDK1 P06493 1/20 0.32
CCNB1 P14635 1/20 0.32
GSK3B P49841 1/20 0.32
CDK5 Q00535 1/20 0.32
CDK5R1 Q15078 1/20 0.32
CCNB3 Q8WWL7 1/20 0.32
METAP1 P53582 1/20 0.32
PTPRC P08575 1/20 0.31
BCL2 P10415 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4409974 1.00 PDK2 (0.40) PDK2S100A4AKR1A1AKR1B1CA1
SCHEMBL6294129 1.00 PDK2 (0.40) PDK2S100A4AKR1A1AKR1B1CA1
SCHEMBL808025 0.91 PDK2 (0.49) PDK2S100A4AKR1A1AKR1B1TDP2
SCHEMBL15138225 0.91 PDK2 (0.49) PDK2S100A4AKR1A1AKR1B1TDP2
SCHEMBL6864497 0.87 TDP2 (0.41) TDP2
SCHEMBL29404184 0.87 PDK2 (0.47) PDK2S100A4AKR1A1AKR1B1CA1
SCHEMBL437007 0.87 PDK2 (0.47) PDK2S100A4AKR1A1AKR1B1CA1
SCHEMBL15138218 0.86 PDK2 (0.41) PDK2AKR1A1AKR1B1PTPRC
SCHEMBL30113034 0.84 PDK2 (0.38) PDK2S100A4AKR1A1AKR1B1CA1
SCHEMBL10020319 0.84 PDK2 (0.38) PDK2S100A4AKR1A1AKR1B1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015049031-A1 HOLE TRANSPORT MATERIAL MERCK PATENT GMBH (DE) 2015-04-09 WO disclosed