SCHEMBL6294129

SCHEMBL6294129

Brc1ccc2c(c1)C1(c3cc(I)ccc3-2)c2cc(I)ccc2-c2ccc(I)cc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.40
S100A4 P26447 1/20 0.35
AKR1A1 P14550 1/20 0.35
AKR1B1 P15121 1/20 0.35
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA4 P22748 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
TDP2 O95551 3/20 0.34
CCNB2 O95067 1/20 0.32
CDK1 P06493 1/20 0.32
CCNB1 P14635 1/20 0.32
GSK3B P49841 1/20 0.32
CDK5 Q00535 1/20 0.32
CDK5R1 Q15078 1/20 0.32
CCNB3 Q8WWL7 1/20 0.32
METAP1 P53582 1/20 0.32
PTPRC P08575 1/20 0.31
BCL2 P10415 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4409974 1.00 PDK2 (0.40) PDK2S100A4AKR1A1AKR1B1CA1
SCHEMBL16625694 1.00 PDK2 (0.40) PDK2S100A4AKR1A1AKR1B1CA1
SCHEMBL808025 0.91 PDK2 (0.49) PDK2S100A4AKR1A1AKR1B1TDP2
SCHEMBL15138225 0.91 PDK2 (0.49) PDK2S100A4AKR1A1AKR1B1TDP2
SCHEMBL6864497 0.87 TDP2 (0.41) TDP2
SCHEMBL29404184 0.87 PDK2 (0.47) PDK2S100A4AKR1A1AKR1B1CA1
SCHEMBL437007 0.87 PDK2 (0.47) PDK2S100A4AKR1A1AKR1B1CA1
SCHEMBL15138218 0.86 PDK2 (0.41) PDK2AKR1A1AKR1B1PTPRC
SCHEMBL30113034 0.84 PDK2 (0.38) PDK2S100A4AKR1A1AKR1B1CA1
SCHEMBL10020319 0.84 PDK2 (0.38) PDK2S100A4AKR1A1AKR1B1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6861567-B2 Spiro compounds, and their use COVION ORGANIC SEMICONDUCTORS GMBH (DE) 2005-03-01 US disclosed
EP-1053216-B1 SPIRANS AND THE USE THEREOF COVION ORGANIC SEMICONDUCTORS (DE) 2003-09-10 EP disclosed
US-20030065190-A1 Spiro compounds, and their use MERCK OLED MATERIALS GMBH (DE) 2003-04-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030065190-A1 Spiro compounds, and their use PKD1, REN, NR3C2 PDK2 756/4885S100A4 2405/4885AKR1A1 38/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.