SCHEMBL16626425

SCHEMBL16626425

CNCc1cn(S(=O)(=O)c2cccnc2)c2cc(Nc3ccc(Cl)cc3C#N)ccc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 6/20 0.39
SLC22A12 Q96S37 1/20 0.35
IDE P14735 1/20 0.35
SCN9A Q15858 1/20 0.35
CYP11B2 P19099 2/20 0.34
CYP11B1 P15538 1/20 0.34
MAOA P21397 1/20 0.34
SRC P12931 1/20 0.34
HTT P42858 1/20 0.34
IMPDH2 P12268 1/20 0.34
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
FBP1 P09467 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
NAMPT P43490 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL16618783 0.99 HTR6 (0.38) HTR6SLC22A12IDESCN9ACYP11B2
SCHEMBL16626428 0.90 HTR6 (0.41) HTR6IDEHTTPDE4APDE4B
Hydrochloric Acid SCHEMBL16619520 0.89 HTR6 (0.40) HTR6IDEHTTPDE4APDE4B
SCHEMBL17971521 0.89 HTR6 (0.40) HTR6IDEHTTPDE4APDE4B
Hydrochloric Acid SCHEMBL16619669 0.89 HTR6 (0.40) HTR6IDEHTTPDE4APDE4B
SCHEMBL16626422 0.89 HTT (0.44) HTR6IDEHTTPDE4APDE4B
Hydrochloric Acid SCHEMBL16618673 0.88 HTT (0.43) HTR6IDEHTTPDE4APDE4B
SCHEMBL16626671 0.87 HTR6 (0.41) HTR6IDEHTTPDE4APDE4B
SCHEMBL16626435 0.87 LRRK2 (0.39) HTR6IDESRCPDE4APDE4B
Hydrochloric Acid SCHEMBL16618624 0.86 HTR6 (0.41) HTR6IDEHTTPDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3052484-B1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAE WOONG PHARMA (KR) 2018-03-21 EP claimed
EP-3052484-B1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAE WOONG PHARMA (KR) 2018-03-21 EP disclosed
US-9676714-B2 Sulfonylindole derivatives and method for preparing the same DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2017-06-13 US disclosed
US-9676714-B2 Sulfonylindole derivatives and method for preparing the same DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2017-06-13 US disclosed
US-20160221946-A1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2016-08-04 US disclosed
US-20160221946-A1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2016-08-04 US disclosed
WO-2015050412-A1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2015-04-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160221946-A1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME GIPR, PGC, SI HTR6 166/4885SLC22A12 3163/4885IDE 2586/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.