SCHEMBL16626446

SCHEMBL16626446

CNCc1cn(S(=O)(=O)c2cccnc2)c2cc(Nc3ccc(F)c(C)c3C)ccc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDE P14735 1/20 0.36
HTR6 P50406 7/20 0.35
HTT P42858 2/20 0.34
CYP19A1 P11511 1/20 0.33
NAMPT P43490 2/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
POLB P06746 1/20 0.33
TBXAS1 P24557 1/20 0.32
HIF1A Q16665 1/20 0.32
CHRNB2 P17787 1/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA4 P43681 1/20 0.32
MEN1 O00255 1/20 0.32
MAPT P10636 1/20 0.32
PABPC1 P11940 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL16619467 0.99 IDE (0.36) IDEHTR6HTTCYP19A1NAMPT
SCHEMBL16626696 0.91 IDE (0.37) IDEHTR6HTTCYP19A1PDE4A
SCHEMBL16626440 0.90 NAMPT (0.37) IDEHTR6HTTCYP19A1NAMPT
Hydrochloric Acid SCHEMBL16618997 0.90 IDE (0.36) IDEHTR6HTTCYP19A1PDE4A
SCHEMBL16626413 0.90 NAMPT (0.37) IDEHTR6HTTCYP19A1NAMPT
SCHEMBL16626422 0.89 HTT (0.44) IDEHTR6HTTNAMPTPDE4A
Hydrochloric Acid SCHEMBL16618761 0.89 NAMPT (0.37) IDEHTR6HTTCYP19A1NAMPT
Hydrochloric Acid SCHEMBL16619306 0.89 NAMPT (0.37) IDEHTR6HTTCYP19A1NAMPT
SCHEMBL17971527 0.89 MAP2K7 (0.38) IDEHTR6HTTNAMPTPOLB
SCHEMBL16626454 0.89 IDE (0.38) IDEHTR6HTTCYP19A1NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3052484-B1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAE WOONG PHARMA (KR) 2018-03-21 EP claimed
EP-3052484-B1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAE WOONG PHARMA (KR) 2018-03-21 EP disclosed
US-9676714-B2 Sulfonylindole derivatives and method for preparing the same DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2017-06-13 US disclosed
US-9676714-B2 Sulfonylindole derivatives and method for preparing the same DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2017-06-13 US disclosed
US-20160221946-A1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2016-08-04 US disclosed
US-20160221946-A1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2016-08-04 US disclosed
WO-2015050412-A1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2015-04-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160221946-A1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME GIPR, PGC, SI IDE 2586/4885HTR6 166/4885HTT 2200/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.