SCHEMBL16626742

SCHEMBL16626742

CNCc1cn(S(=O)(=O)c2ccc(-c3ccccc3)cc2)c2cc(Nc3ccc(C)cc3F)ccc12

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 13/20 0.42
ALK Q9UM73 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
CYP19A1 P11511 1/20 0.38
TNFSF11 O14788 1/20 0.36
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
SLC1A3 P43003 1/20 0.35
SLC1A2 P43004 1/20 0.35
SLC1A1 P43005 1/20 0.35
PCSK9 Q8NBP7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL16618770 0.99 HTR6 (0.41) HTR6ALKL3MBTL1CYP19A1TNFSF11
SCHEMBL16626603 0.95 HTR6 (0.45) HTR6ALKCYP19A1TNFSF11
Hydrochloric Acid SCHEMBL16618833 0.94 HTR6 (0.44) HTR6ALKCYP19A1TNFSF11
SCHEMBL16626773 0.93 HTR6 (0.43) HTR6ALKL3MBTL1CYP19A1PDE4A
Hydrochloric Acid SCHEMBL16619334 0.92 HTR6 (0.43) HTR6ALKL3MBTL1CYP19A1PDE4A
SCHEMBL16626515 0.89 HTR6 (0.41) HTR6ALKCYP19A1PDE4APDE4B
Hydrochloric Acid SCHEMBL16618829 0.89 HTR6 (0.40) HTR6ALKCYP19A1PDE4APDE4B
SCHEMBL16626514 0.88 HTR6 (0.38) HTR6ALKL3MBTL1CYP19A1TNFSF11
SCHEMBL16626527 0.88 HTR6 (0.42) HTR6ALKL3MBTL1CYP19A1PDE4A
SCHEMBL16626760 0.88 HTR6 (0.36) HTR6ALKCYP19A1TNFSF11PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3052484-B1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAE WOONG PHARMA (KR) 2018-03-21 EP claimed
EP-3052484-B1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAE WOONG PHARMA (KR) 2018-03-21 EP disclosed
US-9676714-B2 Sulfonylindole derivatives and method for preparing the same DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2017-06-13 US disclosed
US-9676714-B2 Sulfonylindole derivatives and method for preparing the same DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2017-06-13 US disclosed
US-20160221946-A1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2016-08-04 US disclosed
US-20160221946-A1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2016-08-04 US disclosed
WO-2015050412-A1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2015-04-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160221946-A1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME GIPR, PGC, SI HTR6 166/4885ALK 4825/4885L3MBTL1 4820/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.