SCHEMBL1662676

SCHEMBL1662676

O=C(O)c1nn2ccccc2c1C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHB3 P54753 1/20 0.39
ALDH1A1 P00352 3/20 0.38
CYP2C9 P11712 2/20 0.38
MIF P14174 2/20 0.38
TSHR P16473 2/20 0.38
PDE4B Q07343 2/20 0.38
MEN1 O00255 1/20 0.38
PDE5A O76074 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
PDE4A P27815 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
CYP2C19 P33261 1/20 0.38
BLM P54132 1/20 0.38
KMT2A Q03164 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
PDE3B Q13370 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4917986 0.79 HTR2A (0.44) EPHB3ALDH1A1CYP2C9MIFTSHR
SCHEMBL2809874 0.77 ALDH1A1 (0.49) EPHB3ALDH1A1CYP2C9MIFTSHR
SCHEMBL4917094 0.76 HTR2A (0.45) EPHB3ALDH1A1CYP2C9MIFTSHR
SCHEMBL35264 0.76 PTGS1 (0.45) EPHB3ALDH1A1CYP2C9MIFTSHR
SCHEMBL12686677 0.76 SPR (0.45) ALDH1A1CYP2C9MIFTSHRPDE4B
SCHEMBL16223183 0.75 MIF (0.44) EPHB3ALDH1A1CYP2C9MIFTSHR
SCHEMBL4183274 0.75 EGFR (0.36) EPHB3ALDH1A1CYP2C9MIFTSHR
SCHEMBL5133264 0.74 APOBEC3A (0.45) ALDH1A1MEN1KMT2AELANEHPGD
SCHEMBL1665454 0.73 EGFR (0.40) EPHB3ALDH1A1CYP2C9MIFTSHR
SCHEMBL35212140 0.72 MIF (0.41) EPHB3ALDH1A1CYP2C9MIFTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011050284-A1 PYRAZOLYLPYRIDINE ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2011-04-28 WO disclosed