SCHEMBL16627593

SCHEMBL16627593

O=C(NCCc1ccc(Br)cc1)c1cc2ccccc2[nH]c1=O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.51
ALDH1A1 P00352 1/20 0.51
KMT2A Q03164 2/20 0.50
TNKS O95271 1/20 0.49
TNKS2 Q9H2K2 1/20 0.49
SMYD3 Q9H7B4 2/20 0.49
NPC1 O15118 3/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
RAB9A P51151 2/20 0.47
MEN1 O00255 1/20 0.47
PKM P14618 1/20 0.47
CNR2 P34972 2/20 0.46
TP53 P04637 1/20 0.46
MAPT P10636 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA4 P22748 1/20 0.44
CA5A P35218 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL34468791 0.90 KDM4E (0.62) KDM4EALDH1A1KMT2ASMYD3NPC1
SCHEMBL16627891 0.89 KDM4E (0.52) KDM4EALDH1A1KMT2ASMYD3NPC1
SCHEMBL16627713 0.88 CNR2 (0.59) KDM4EALDH1A1KMT2ASMYD3NPC1
SCHEMBL16627831 0.88 KDM4E (0.51) KDM4EALDH1A1KMT2ASMYD3NPC1
SCHEMBL16627739 0.87 SMYD3 (0.50) KDM4EALDH1A1KMT2ASMYD3NPC1
SCHEMBL16627887 0.85 KDM4E (0.48) KDM4EALDH1A1KMT2ASMYD3NPC1
SCHEMBL34468766 0.84 SMYD3 (0.49) KDM4EALDH1A1KMT2ASMYD3NPC1
SCHEMBL16627868 0.84 KDM4E (0.48) KDM4EALDH1A1KMT2ASMYD3NPC1
SCHEMBL16627706 0.82 ALDH1A1 (0.51) KDM4EALDH1A1KMT2ANPC1RAB9A
SCHEMBL34468807 0.81 PARP1 (0.50) KDM4EALDH1A1KMT2ASMYD3NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015050379-A1 NOVEL QUINOLINONE DERIVATIVE AND USE THEREOF 광주과학기술원 2015-04-09 WO disclosed