SCHEMBL1662762

SCHEMBL1662762

C(#Cc1ncc(CCN2CCOCC2)s1)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.46
SIGMAR1 Q99720 1/20 0.46
GRM5 P41594 8/20 0.46
KMT2A Q03164 2/20 0.43
HTT P42858 1/20 0.43
ALDH1A1 P00352 1/20 0.42
MEN1 O00255 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
LTA4H P09960 1/20 0.40
GAA P10253 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1662778 0.90 GRM5 (0.51) SIGMAR1GRM5LTA4H
SCHEMBL1658169 0.87 SMN1; SMN2 (0.52) GRM5KMT2AHTTALDH1A1MEN1
SCHEMBL1657728 0.76 GRM5 (0.53) GRM5KMT2AALDH1A1MEN1LTA4H
SCHEMBL1659965 0.76 GRM5 (0.50) GRM5KMT2AHTTALDH1A1GAA
SCHEMBL1657377 0.76 ALDH1A1 (0.49) GRM5KMT2AALDH1A1NPC1RAB9A
SCHEMBL1663193 0.76 GRM5 (0.45) GRM5
SCHEMBL1657724 0.75 GRM5 (0.55) GRM5KMT2AALDH1A1MEN1GAA
SCHEMBL1658480 0.75 GRM5 (0.45) GRM5KMT2AHTTALDH1A1GAA
SCHEMBL1663726 0.72 GRM5 (0.47) GRM5
SCHEMBL1659148 0.72 ALDH1A1 (0.56) GRM5KMT2AHTTALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2490541-A1 2-SUBSTITUTED-ETHYNYLTHIAZOLE DERIVATIVES AND USES OF SAME H. Lundbeck A/S (DK) 2012-08-29 EP claimed
WO-2011050063-A1 2-SUBSTITUTED-ETHYNYLTHIAZOLE DERIVATIVES AND USES OF SAME H. LUNDBECK A/S (DK) 2011-04-28 WO claimed