SCHEMBL16627627

SCHEMBL16627627

COc1ccc(Cn2c(=O)ccc3c(NC(=O)C4(C)CC5CC(C)(C)CC(C)(C5)C4)cccc32)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 10/20 0.51
P2RX4 Q99571 1/20 0.41
HDAC1 Q13547 2/20 0.40
ALDH1A1 P00352 2/20 0.37
GAA P10253 1/20 0.37
HDAC11 Q96DB2 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
LMNA P02545 1/20 0.37
PDE1A P54750 1/20 0.36
PDE1B Q01064 1/20 0.36
PDE1C Q14123 1/20 0.36
MAPT P10636 3/20 0.36
KDM4E B2RXH2 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
MAPK1 P28482 1/20 0.35
PTGER3 P43115 1/20 0.35
RECQL P46063 1/20 0.35
TP53 P04637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16627629 0.88 P2RX7 (0.60) P2RX7P2RX4HDAC1ALDH1A1HDAC11
SCHEMBL16627867 0.88 P2RX7 (0.52) P2RX7P2RX4HDAC1ALDH1A1GAA
SCHEMBL16627862 0.82 P2RX7 (0.51) P2RX7P2RX4HDAC1ALDH1A1HDAC11
SCHEMBL16627913 0.80 P2RX7 (0.52) P2RX7P2RX4HDAC1HDAC11HDAC8
SCHEMBL16627628 0.78 P2RX7 (0.67) P2RX7P2RX4HDAC1HDAC11HDAC8
SCHEMBL16627863 0.78 P2RX7 (0.49) P2RX7P2RX4HDAC1ALDH1A1HDAC11
SCHEMBL16627910 0.77 P2RX7 (0.58) P2RX7P2RX4HDAC1LMNAMAPT
SCHEMBL16627911 0.76 P2RX7 (0.51) P2RX7P2RX4HDAC1HDAC11HDAC8
SCHEMBL16627866 0.75 P2RX7 (0.49) P2RX7P2RX4HDAC1HDAC11HDAC8
SCHEMBL16627793 0.75 P2RX7 (0.80) P2RX7P2RX4HDAC1HDAC11HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015050379-A1 NOVEL QUINOLINONE DERIVATIVE AND USE THEREOF 광주과학기술원 2015-04-09 WO disclosed