SCHEMBL16627863

SCHEMBL16627863

COc1ccc(Cn2c(=O)ccc3c(NNC(=O)C4(C)CC5CC(CC(C)(Cl)C5)C4)cccc32)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 13/20 0.49
P2RX4 Q99571 1/20 0.39
HDAC1 Q13547 2/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
LMNA P02545 2/20 0.37
PDE1A P54750 1/20 0.36
PDE1B Q01064 1/20 0.36
PDE1C Q14123 1/20 0.36
ALDH1A1 P00352 1/20 0.36
NPC1 O15118 1/20 0.35
TP53 P04637 1/20 0.35
POLB P06746 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
NFKB1 P19838 1/20 0.35
HTT P42858 1/20 0.35
RAB9A P51151 1/20 0.35
NFKB2 Q00653 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16627913 0.94 P2RX7 (0.52) P2RX7P2RX4HDAC1HDAC11HDAC8
SCHEMBL16627866 0.93 P2RX7 (0.49) P2RX7P2RX4HDAC1HDAC11HDAC8
SCHEMBL16627911 0.92 P2RX7 (0.51) P2RX7P2RX4HDAC1HDAC11HDAC8
SCHEMBL16627629 0.85 P2RX7 (0.60) P2RX7P2RX4HDAC1HDAC11HDAC8
SCHEMBL16627910 0.84 P2RX7 (0.58) P2RX7P2RX4HDAC1LMNATP53
SCHEMBL16627865 0.79 P2RX7 (0.58) P2RX7P2RX4
SCHEMBL16627862 0.78 P2RX7 (0.51) P2RX7P2RX4HDAC1HDAC11HDAC8
SCHEMBL16627627 0.78 P2RX7 (0.51) P2RX7P2RX4HDAC1HDAC11HDAC8
SCHEMBL16627717 0.76 P2RX7 (0.48) P2RX7P2RX4HDAC1HDAC11HDAC8
SCHEMBL16627673 0.76 P2RX7 (0.48) P2RX7P2RX4HDAC1HDAC11HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015050379-A1 NOVEL QUINOLINONE DERIVATIVE AND USE THEREOF 광주과학기술원 2015-04-09 WO disclosed