SCHEMBL16627765

SCHEMBL16627765

C=C(C)c1cc2ccccc2n(CC)c1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.47
CASP1 P29466 1/20 0.47
CASP7 P55210 1/20 0.47
CNR1 P21554 6/20 0.44
CNR2 P34972 6/20 0.44
KDM4E B2RXH2 5/20 0.43
ALDH1A1 P00352 3/20 0.43
LMNA P02545 1/20 0.43
HPGD P15428 1/20 0.43
HSD17B10 Q99714 1/20 0.43
CA12 O43570 1/20 0.43
CA9 Q16790 1/20 0.43
RCE1 Q9Y256 1/20 0.42
DAO P14920 1/20 0.41
CCR2 P41597 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
TP53 P04637 1/20 0.40
SRC P12931 1/20 0.39
MAPT P10636 1/20 0.39
RECQL P46063 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16627568 0.84 CA12 (0.51) MAPK1CASP1CASP7CNR1CNR2
SCHEMBL6547150 0.82 MAPK1 (0.47) MAPK1CASP1CASP7CNR1CNR2
SCHEMBL16627889 0.78 L3MBTL1 (0.41) MAPK1CNR1CNR2KDM4ELMNA
SCHEMBL11824046 0.78 DAO (0.62) MAPK1CASP1CASP7KDM4EALDH1A1
SCHEMBL16627741 0.77 AHR (0.61) CNR1CNR2ALDH1A1TP53MAPT
SCHEMBL434663 0.77 KDM4E (0.50) MAPK1CASP1CASP7KDM4EALDH1A1
SCHEMBL16627569 0.75 CNR1 (0.60) MAPK1CNR1CNR2KDM4EALDH1A1
SCHEMBL30355091 0.74 BTK (0.48) MAPK1CASP1CASP7KDM4EALDH1A1
SCHEMBL26620879 0.74 KDM4E (0.47) MAPK1CASP1CASP7KDM4EALDH1A1
SCHEMBL28325706 0.74 LMNA (0.48) MAPK1CASP1CASP7KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015050379-A1 NOVEL QUINOLINONE DERIVATIVE AND USE THEREOF 광주과학기술원 2015-04-09 WO disclosed