SCHEMBL16627794

SCHEMBL16627794

COC(=O)c1cc2c(NC(=O)C3(C)CC4CC(CC(C)(Br)C4)C3)cccc2n(Cc2ccc(OC)cc2)c1=O

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 10/20 0.77
HDAC1 Q13547 2/20 0.40
P2RX4 Q99571 1/20 0.39
MAPK8 P45983 1/20 0.39
PDE1B Q01064 2/20 0.38
PDE1C Q14123 2/20 0.38
PDE1A P54750 1/20 0.38
MAPT P10636 2/20 0.38
HDAC11 Q96DB2 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
TP53 P04637 2/20 0.37
RXFP1 Q9HBX9 1/20 0.37
NPC1 O15118 1/20 0.37
LMNA P02545 1/20 0.37
POLB P06746 1/20 0.37
HPGD P15428 1/20 0.37
TSHR P16473 1/20 0.37
NFKB1 P19838 1/20 0.37
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16627793 0.94 P2RX7 (0.80) P2RX7HDAC1P2RX4MAPK8PDE1B
SCHEMBL16627901 0.90 P2RX7 (0.78) P2RX7HDAC1P2RX4MAPK8MAPT
SCHEMBL16627903 0.84 P2RX7 (0.81) P2RX7HDAC1P2RX4MAPTTP53
SCHEMBL16627629 0.81 P2RX7 (0.60) P2RX7HDAC1P2RX4PDE1BPDE1C
SCHEMBL16627902 0.80 P2RX7 (1.00) P2RX7HDAC1P2RX4TP53NPC1
SCHEMBL16627866 0.78 P2RX7 (0.49) P2RX7HDAC1P2RX4MAPK8HDAC11
SCHEMBL16627612 0.78 P2RX7 (1.00) P2RX7P2RX4LMNA
SCHEMBL16627791 0.77 P2RX7 (0.69) P2RX7HDAC1P2RX4MAPK8MAPT
SCHEMBL16627607 0.77 P2RX7 (0.79) P2RX7MAPK8MAPTTP53RXFP1
SCHEMBL16627907 0.76 P2RX7 (0.79) P2RX7HDAC1P2RX4MAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015050379-A1 NOVEL QUINOLINONE DERIVATIVE AND USE THEREOF 광주과학기술원 2015-04-09 WO disclosed