SCHEMBL16627902

SCHEMBL16627902

COC(=O)c1cc2c(NC(=O)C3CCCCC3)cccc2n(Cc2ccc(OC)cc2)c1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 10/20 1.00
HPGD P15428 3/20 0.47
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 3/20 0.47
HSD17B10 Q99714 3/20 0.47
NPSR1 Q6W5P4 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
LMNA P02545 2/20 0.47
HTT P42858 2/20 0.47
NPC1 O15118 1/20 0.47
TP53 P04637 1/20 0.47
POLB P06746 1/20 0.47
TSHR P16473 1/20 0.47
NFKB1 P19838 1/20 0.47
RAB9A P51151 1/20 0.47
NFKB2 Q00653 1/20 0.47
RELA Q04206 1/20 0.47
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16627789 0.85 P2RX7 (0.83) P2RX7HPGDKDM4EALDH1A1HSD17B10
SCHEMBL16627791 0.82 P2RX7 (0.69) P2RX7NPC1TP53RAB9AP2RX4
SCHEMBL16627793 0.81 P2RX7 (0.80) P2RX7HPGDSMN1; SMN2LMNAHTT
SCHEMBL16627790 0.80 P2RX7 (0.70) P2RX7HPGDKDM4EALDH1A1SMN1; SMN2
SCHEMBL16627794 0.80 P2RX7 (0.77) P2RX7HPGDSMN1; SMN2LMNAHTT
SCHEMBL16627903 0.78 P2RX7 (0.81) P2RX7TP53P2RX4HDAC1
SCHEMBL16627901 0.76 P2RX7 (0.78) P2RX7TP53P2RX4HDAC1
SCHEMBL16627607 0.73 P2RX7 (0.79) P2RX7ALDH1A1TP53
SCHEMBL16627907 0.72 P2RX7 (0.79) P2RX7KDM4EHSD17B10SMN1; SMN2NPC1
SCHEMBL16627908 0.72 P2RX7 (0.91) P2RX7TP53P2RX4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015050379-A1 NOVEL QUINOLINONE DERIVATIVE AND USE THEREOF 광주과학기술원 2015-04-09 WO disclosed