SCHEMBL16627673

SCHEMBL16627673

COc1ccc(Cn2c(=O)ccc3c(NNC(=O)CC45CC(C)CC(Cl)(CC(C)C4)C5)cccc32)cc1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 10/20 0.48
HDAC1 Q13547 3/20 0.38
HDAC8 Q9BY41 2/20 0.38
HDAC6 Q9UBN7 2/20 0.38
HDAC11 Q96DB2 1/20 0.38
P2RX4 Q99571 1/20 0.38
MCL1 Q07820 1/20 0.36
MAPT P10636 3/20 0.36
TP53 P04637 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
P2RX3 P56373 1/20 0.35
TRPV1 Q8NER1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16627717 0.92 P2RX7 (0.48) P2RX7HDAC1HDAC8HDAC6HDAC11
SCHEMBL16627667 0.91 P2RX7 (0.47) P2RX7HDAC1HDAC8HDAC6HDAC11
SCHEMBL16627865 0.88 P2RX7 (0.58) P2RX7P2RX4P2RX3
SCHEMBL16627911 0.78 P2RX7 (0.51) P2RX7HDAC1HDAC8HDAC6HDAC11
SCHEMBL16627863 0.76 P2RX7 (0.49) P2RX7HDAC1HDAC8HDAC6HDAC11
SCHEMBL16627913 0.76 P2RX7 (0.52) P2RX7HDAC1HDAC8HDAC6HDAC11
SCHEMBL16627866 0.74 P2RX7 (0.49) P2RX7HDAC1HDAC8HDAC6HDAC11
SCHEMBL16627864 0.74 P2RX7 (0.60) P2RX7HDAC1P2RX4MAPTTP53
SCHEMBL16627628 0.73 P2RX7 (0.67) P2RX7HDAC1HDAC8HDAC6HDAC11
SCHEMBL16627910 0.73 P2RX7 (0.58) P2RX7HDAC1P2RX4MAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015050379-A1 NOVEL QUINOLINONE DERIVATIVE AND USE THEREOF 광주과학기술원 2015-04-09 WO disclosed