SCHEMBL16629095

SCHEMBL16629095

CC(C)(C)c1[nH]c2ccc(I)cc2c1-c1nc2c3cccnc3c3ncccc3c2[nH]1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 3/20 0.35
GSK3B P49841 3/20 0.35
CDK5 Q00535 2/20 0.35
CDK5R1 Q15078 2/20 0.35
CDK4 P11802 1/20 0.34
CCND1 P24385 1/20 0.34
FLT3 P36888 2/20 0.33
CCNB2 O95067 1/20 0.33
CDK1 P06493 1/20 0.33
CCNB1 P14635 1/20 0.33
CCNB3 Q8WWL7 1/20 0.33
PTGES O14684 5/20 0.33
JAK2 O60674 2/20 0.33
PARP1 P09874 2/20 0.33
GABRA1 P14867 2/20 0.32
GABRG2 P18507 2/20 0.32
GABRB3 P28472 2/20 0.32
GABRA5 P31644 2/20 0.32
GABRA3 P34903 2/20 0.32
GABRA2 P47869 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10067290 0.89 CDK4 (0.41) CDK4CCND1PTGESJAK2PARP1
SCHEMBL16624849 0.88 PTGES (0.41) GSK3AGSK3BCDK4CCND1PTGES
SCHEMBL10067287 0.88 KIF11 (0.45) GSK3AGSK3BCDK5CDK4CCND1
SCHEMBL10067297 0.87 PTGES (0.37) GSK3AGSK3BCDK5CDK5R1CDK4
SCHEMBL10067328 0.87 PTGES (0.43) GSK3AGSK3BCDK5CDK5R1CDK4
SCHEMBL10067315 0.86 PTGES (0.40) CDK4CCND1PTGESJAK2GABRA1
SCHEMBL16629721 0.85 KDM4E (0.43) GSK3AGSK3BCDK5CDK5R1CDK4
SCHEMBL10067285 0.85 PTGES (0.41) CDK4CCND1PTGESKDM4EMAPT
SCHEMBL10067300 0.84 CDK4 (0.33) CDK4CCND1PTGESJAK2PARP1
SCHEMBL10082768 0.84 L3MBTL1 (0.41) GSK3AGSK3BCDK5CDK5R1CCNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015051302-A1 COMPOSITIONS AND METHODS FOR TREATING CANCERS APTOSE BIOSCIENCES INC. (CA) 2015-04-09 WO disclosed