SCHEMBL16631329

SCHEMBL16631329

CC(=O)CCc1ccc2c(c1)OCc1cc(COCc3ccccc3)ccc1-2

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 9/20 0.44
AKR1B1 P15121 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MAOA P21397 2/20 0.40
MAOB P27338 2/20 0.40
LTB4R Q15722 1/20 0.40
LTB4R2 Q9NPC1 1/20 0.40
ROCK1 Q13464 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18165301 0.91 AKR1B1 (0.47) ROCK2AKR1B1MAOAMAOBLTB4R
SCHEMBL16631357 0.82 ROCK2 (0.41) ROCK2AKR1B1MAOA
SCHEMBL16631400 0.76 ROCK2 (0.40) ROCK2AKR1B1ROCK1
SCHEMBL17954207 0.74 PRF1 (0.37) ROCK2AKR1B1ROCK1
SCHEMBL18165307 0.74 AKR1B1 (0.47) ROCK2AKR1B1LTB4RLTB4R2
SCHEMBL10898501 0.73 HTR2C (0.54) ALDH1A1MAOA
SCHEMBL18165309 0.72 FFAR1 (0.51) AKR1B1MAOAMAOB
SCHEMBL20216036 0.71 ROCK2 (0.38) ROCK2AKR1B1ROCK1
SCHEMBL22540441 0.71 FFAR1 (0.49) AKR1B1MAOAMAOB
SCHEMBL5657672 0.71 AKR1B1 (0.58) ROCK2AKR1B1LTB4RLTB4R2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015051045-A2 3'END CAPS FOR RNAi AGENTS FOR USE IN RNA INTERFERENCE NOVARTIS AG (CH) 2015-04-09 WO disclosed