SCHEMBL16631357

SCHEMBL16631357

CC(=O)CCc1ccc2c(c1)OCc1cc(CN)ccc1-2

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 8/20 0.41
AKR1B1 P15121 1/20 0.40
AAK1 Q2M2I8 2/20 0.38
KCNJ1 P48048 1/20 0.38
KCNH2 Q12809 1/20 0.38
KDM4E B2RXH2 1/20 0.37
NPC1 O15118 1/20 0.37
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
MAPT P10636 1/20 0.37
MAOA P21397 1/20 0.37
SLC6A2 P23975 1/20 0.37
RAB9A P51151 1/20 0.37
SLC6A3 Q01959 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16631329 0.82 ROCK2 (0.44) ROCK2AKR1B1MAOA
SCHEMBL18165307 0.77 AKR1B1 (0.47) ROCK2AKR1B1AAK1KCNJ1KCNH2
SCHEMBL803505 0.75 KCNJ1 (0.43) ROCK2AKR1B1AAK1KCNJ1KCNH2
SCHEMBL16631067 0.74 ITGB3 (0.46) MAOA
SCHEMBL10898501 0.73 HTR2C (0.54) KDM4ENPC1LMNATP53CYP1A2
SCHEMBL4469820 0.72 ROCK2 (0.51) ROCK2
SCHEMBL9980133 0.72 PARP1 (0.44) ROCK2AKR1B1AAK1KCNJ1KCNH2
SCHEMBL10899522 0.72 RAB9A (0.47) KDM4ENPC1LMNATP53CYP1A2
SCHEMBL18165301 0.71 AKR1B1 (0.47) ROCK2AKR1B1MAOA
SCHEMBL10897771 0.70 HSD17B1 (0.58) AKR1B1KDM4ENPC1LMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015051045-A2 3'END CAPS FOR RNAi AGENTS FOR USE IN RNA INTERFERENCE NOVARTIS AG (CH) 2015-04-09 WO disclosed