SCHEMBL16631512

SCHEMBL16631512

CCc1ccc2c(c1)OCc1cc(COC(=O)CCC(=O)O)ccc1-2

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.41
ROCK2 O75116 6/20 0.40
CYP3A4 P08684 1/20 0.39
AAK1 Q2M2I8 5/20 0.39
FAAH O00519 1/20 0.39
MGLL Q99685 1/20 0.39
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16631400 0.93 ROCK2 (0.40) AKR1B1ROCK2CYP3A4AAK1FAAH
SCHEMBL16624802 0.80 ROCK2 (0.41) AKR1B1ROCK2AAK1FAAHMGLL
SCHEMBL9980133 0.79 PARP1 (0.44) AKR1B1ROCK2AAK1GAAMAPT
SCHEMBL16624806 0.76 ROCK2 (0.38) AKR1B1ROCK2CYP3A4MAPT
SCHEMBL17954212 0.75 AKR1B1 (0.40) AKR1B1ROCK2AAK1GAAMAPT
SCHEMBL18165301 0.74 AKR1B1 (0.47) AKR1B1ROCK2
SCHEMBL16624619 0.73 MAOA (0.41) ROCK2
SCHEMBL17954207 0.73 PRF1 (0.37) AKR1B1ROCK2GAAMAPT
SCHEMBL18165307 0.72 AKR1B1 (0.47) AKR1B1ROCK2AAK1
SCHEMBL18462572 0.71 ROCK2 (0.42) AKR1B1ROCK2AAK1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015051045-A2 3'END CAPS FOR RNAi AGENTS FOR USE IN RNA INTERFERENCE NOVARTIS AG (CH) 2015-04-09 WO disclosed