SCHEMBL16634909

SCHEMBL16634909

CCCC(=O)Nc1ccc2cnccc2c1

nearest known ligand 0.61

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PRMT3 O60678 6/20 0.61
IMPDH2 P12268 5/20 0.60
NOTUM Q6P988 5/20 0.59
SMN1; SMN2 Q16637 2/20 0.55
NPC1 O15118 1/20 0.55
LMNA P02545 1/20 0.55
RAB9A P51151 1/20 0.55
KDM4E B2RXH2 2/20 0.54
ALDH1A1 P00352 2/20 0.54
AAK1 Q2M2I8 1/20 0.54
HPGD P15428 1/20 0.53
HSD17B10 Q99714 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12201798 0.88 PRMT3 (0.64) PRMT3IMPDH2NOTUM
Hydrochloric Acid SCHEMBL111600 0.87 PRMT3 (0.62) PRMT3IMPDH2NOTUM
SCHEMBL21430054 0.86 IMPDH2 (0.62) PRMT3IMPDH2NOTUM
SCHEMBL30176801 0.84 KDM4E (0.66) PRMT3IMPDH2NOTUMKDM4EALDH1A1
SCHEMBL20262924 0.84 KDM4E (0.66) PRMT3IMPDH2NOTUMKDM4EALDH1A1
SCHEMBL19860095 0.84 IMPDH2 (0.62) PRMT3IMPDH2NOTUM
SCHEMBL19860105 0.83 PRMT3 (0.62) PRMT3IMPDH2NOTUM
SCHEMBL2162755 0.82 NOTUM (0.62) PRMT3IMPDH2NOTUM
SCHEMBL12201759 0.82 IMPDH2 (0.61) PRMT3IMPDH2NOTUM
SCHEMBL19860096 0.82 NOTUM (0.65) PRMT3IMPDH2NOTUMSMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9890123-B2 6-aminoisoquinoline compounds AERIE PHARMACEUTICALS, INC. (US) 2018-02-13 US disclosed
EP-3055304-A1 NOVEL PYRIDYLOXYACETYL TETRAHYDROISOQUINOLINE COMPOUNDS USEFUL AS NAMPT INHIBITORS Eli Lilly and Company (US) 2016-08-17 EP disclosed
WO-2015054060-A1 NOVEL PYRIDYLOXYACETYL TETRAHYDROISOQUINOLINE COMPOUNDS USEFUL AS NAMPT INHIBITORS ELI LILLY AND COMPANY (US) 2015-04-16 WO disclosed