SCHEMBL16637355

SCHEMBL16637355

CCOC(=O)c1cc(N)cc(C(F)(F)F)c1F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.47
IDO1 P14902 1/20 0.43
ALDH1A1 P00352 4/20 0.43
HSD17B10 Q99714 2/20 0.43
GAA P10253 2/20 0.42
MAPK1 P28482 1/20 0.42
LMNA P02545 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAOA P21397 1/20 0.41
TSHR P16473 1/20 0.41
NPC1 O15118 3/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
MAPT P10636 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
ALOX15 P16050 1/20 0.41
HDAC3 O15379 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7593446 0.83 TSHR (0.44) KDM4EIDO1ALDH1A1LMNAL3MBTL1
SCHEMBL29945861 0.82 KDM4E (0.33) KDM4EIDO1ALDH1A1GAAL3MBTL1
SCHEMBL16637855 0.82 NOTUM (0.43) KDM4EIDO1ALDH1A1LMNAL3MBTL1
SCHEMBL23526137 0.82 KDM4E (0.33) KDM4EIDO1ALDH1A1GAAL3MBTL1
SCHEMBL16638001 0.78 NPC1 (0.48) ALDH1A1LMNAL3MBTL1NPC1MEN1
SCHEMBL23326804 0.78 KIF11 (0.38) KDM4EALDH1A1HSD17B10GAATSHR
SCHEMBL16647668 0.77 KDM4E (0.47) KDM4EIDO1ALDH1A1HSD17B10GAA
SCHEMBL16529867 0.76 KDM4E (0.44) KDM4EIDO1ALDH1A1HSD17B10GAA
SCHEMBL24566862 0.76 KDM4E (0.43) KDM4EALDH1A1HSD17B10GAACYP3A4
SCHEMBL24566864 0.75 HDAC4 (0.34) ALDH1A1GAALMNATSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015051496-A1 ANTIDIABETIC TRICYCLIC COMPOUNDS MERCK SHARP & DOHME CORP. (US) 2015-04-16 WO disclosed