SCHEMBL16638382

SCHEMBL16638382

COc1cc(-c2nc3cccc(C(=O)O)c3[nH]2)cc(OC)c1-c1ccccc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 3/20 0.70
CYP1A1 P04798 2/20 0.46
CYP1B1 Q16678 2/20 0.46
CYP1A2 P05177 1/20 0.46
GUSB P08236 2/20 0.46
FABP3 P05413 1/20 0.45
FABP4 P15090 1/20 0.45
FABP5 Q01469 1/20 0.45
PARP1 P09874 3/20 0.45
SMPD3 Q9NY59 3/20 0.44
NOX1 Q9Y5S8 1/20 0.44
KMT2A Q03164 1/20 0.44
PDE10A Q9Y233 1/20 0.44
KDM4E B2RXH2 2/20 0.43
NPC1 O15118 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4740751 0.87 GUSB (0.59) DHODHCYP1A1CYP1B1CYP1A2GUSB
SCHEMBL696548 0.83 DHODH (0.56) DHODHCYP1A2PARP1KMT2AKDM4E
SCHEMBL505197 0.82 DHODH (1.00) DHODHPARP1
SCHEMBL28116288 0.81 PARP1 (0.53) DHODHCYP1A1CYP1B1CYP1A2GUSB
SCHEMBL505569 0.80 DHODH (0.55) DHODHPARP1KDM4ENPC1ALDH1A1
SCHEMBL504921 0.78 DHODH (0.67) DHODHKMT2AKDM4ENPC1ALDH1A1
SCHEMBL697780 0.77 KDM4E (0.54) DHODHGUSBPARP1KMT2AKDM4E
SCHEMBL10211823 0.76 DHODH (0.64) DHODHFABP3FABP4FABP5KMT2A
SCHEMBL6840289 0.76 PIN1 (0.56) DHODHPARP1KMT2AKDM4ENPC1
SCHEMBL505582 0.76 DHODH (0.64) DHODHPARP1KMT2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9006454-B2 Dihydroorotate dehydrogenase inhibitors MERCK SERONO S.A. (CH) 2015-04-14 US disclosed
US-9006454-B2 Dihydroorotate dehydrogenase inhibitors MERCK SERONO S.A. (CH) 2015-04-14 US disclosed