SCHEMBL16638715

SCHEMBL16638715

COc1cc(Cl)cc(Nc2ncccc2C=O)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 6/20 0.44
KMT2A Q03164 6/20 0.44
HTT P42858 3/20 0.44
PKM P14618 1/20 0.44
MAPK1 P28482 1/20 0.44
NPC1 O15118 2/20 0.41
ALDH1A1 P00352 2/20 0.41
RAB9A P51151 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
MAPT P10636 4/20 0.41
PIK3C2B O00750 1/20 0.41
PIK3C2G O75747 1/20 0.41
TUBB4A P04350 1/20 0.40
TUBB P07437 1/20 0.40
TUBA3C P0DPH7 1/20 0.40
TUBA1B P68363 1/20 0.40
TUBA4A P68366 1/20 0.40
TUBB4B P68371 1/20 0.40
TUBB3 Q13509 1/20 0.40
TUBB2A Q13885 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8835541 0.87 GRM4 (0.50) MEN1KMT2AHTTNPC1ALDH1A1
SCHEMBL9402386 0.83 MEN1 (0.63) MEN1KMT2AHTTPKMMAPK1
SCHEMBL8835483 0.81 RAB9A (0.60) MEN1KMT2AHTTMAPK1NPC1
SCHEMBL15636276 0.79 MEN1 (0.72) MEN1KMT2AHTTPKMMAPK1
SCHEMBL17363143 0.79 MEN1 (0.58) MEN1KMT2AHTTPKMMAPK1
SCHEMBL16638716 0.79 MEN1 (0.58) MEN1KMT2AHTTPKMMAPK1
SCHEMBL6643061 0.79 NPC1 (0.59) MEN1KMT2AHTTNPC1ALDH1A1
SCHEMBL10680055 0.78 TEK (0.50) ALDH1A1RAB9ATUBB1GAAEGFR
SCHEMBL16638713 0.78 GRM4 (0.58) MEN1KMT2ANPC1ALDH1A1RAB9A
SCHEMBL9402383 0.77 RAB9A (0.57) MEN1KMT2AHTTNPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9006451-B1 2-anilinonicotinyl based chalcones useful as potential anticancer agents and process for preparation thereof COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2015-04-14 US disclosed