SCHEMBL16638817

SCHEMBL16638817

CC[C@@H](COC)NC(=O)OC(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSK P43235 8/20 0.45
CTSS P25774 4/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA7 P43166 1/20 0.45
SYK P43405 2/20 0.44
TAS1R3 Q7RTX0 3/20 0.42
TAS1R1 Q7RTX1 3/20 0.42
TAS1R2 Q8TE23 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
CYP2D6 P10635 1/20 0.41
ATM Q13315 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3389057 0.91 CA1 (0.49) CTSKCTSSCA1CA2CA7
SCHEMBL9911449 0.87 CA1 (0.52) CTSKCTSSCA1CA2CA7
SCHEMBL1987512 0.86 CA1 (0.45) CTSKCTSSCA1CA2CA7
SCHEMBL1987513 0.86 CA1 (0.45) CTSKCTSSCA1CA2CA7
SCHEMBL6401398 0.86 CA1 (0.45) CTSKCTSSCA1CA2CA7
SCHEMBL23605451 0.84 CA1 (0.44) CTSKCTSSCA1CA2CA7
SCHEMBL15541356 0.84 CA1 (0.44) CTSKCTSSCA1CA2CA7
SCHEMBL20886481 0.84 CA1 (0.44) CTSKCTSSCA1CA2CA7
SCHEMBL15968312 0.84 CA1 (0.44) CTSKCTSSCA1CA2CA7
SCHEMBL1988335 0.84 CA1 (0.44) CTSKCTSSCA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180079727-A1 9-MEMBERED FUSED RING DERIVATIVE SHIONOGI & CO., LTD. (JP) 2018-03-22 US disclosed
EP-2540720-B1 1,3,4,8-TETRAHYDRO-2H-PYRIDO[1,2-A]PYRAZINE DERIVATIVE AND USE OF SAME AS HIV INTEGRASE INHIBITOR JAPAN TOBACCO INC (JP) 2015-04-15 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180079727-A1 9-MEMBERED FUSED RING DERIVATIVE ACSS2, AGTR2, ACSL3 CTSK 2427/4885CTSS 1021/4885CA1 1525/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.