SCHEMBL16638841

SCHEMBL16638841

COc1nccc(-c2ccccc2)c1I

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.49
MAPT P10636 3/20 0.49
NPC1 O15118 3/20 0.49
RAB9A P51151 3/20 0.49
MEN1 O00255 2/20 0.49
ALDH1A1 P00352 2/20 0.49
CRHBP P24387 1/20 0.49
CRHR2 Q13324 1/20 0.49
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
SQOR Q9Y6N5 3/20 0.44
CASP1 P29466 1/20 0.40
CHEK1 O14757 1/20 0.38
CCNA2 P20248 1/20 0.38
CDK2 P24941 1/20 0.38
IKBKB O14920 1/20 0.38
CHUK O15111 1/20 0.38
DAPK3 O43293 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28635180 0.80 KMT2A (0.50) KMT2AMAPTNPC1RAB9AMEN1
SCHEMBL13144468 0.80 SQOR (0.57) KMT2AMAPTNPC1RAB9AMEN1
SCHEMBL13422264 0.76 DHODH (0.53) KMT2AMAPTNPC1RAB9AMEN1
SCHEMBL24457916 0.75 CCR1 (0.37) KMT2AMAPTNPC1RAB9AMEN1
SCHEMBL29956027 0.75 KMT2A (0.46) KMT2AMAPTNPC1RAB9AMEN1
SCHEMBL12960812 0.75 KMT2A (0.46) KMT2AMAPTNPC1RAB9AMEN1
SCHEMBL29223019 0.73 MAPT (0.45) KMT2AMAPTNPC1RAB9AMEN1
SCHEMBL4056518 0.73 DHODH (0.54) KMT2AMAPTNPC1RAB9AMEN1
SCHEMBL13752829 0.72 GABRA1 (0.50) KMT2AMAPTNPC1RAB9AMEN1
SCHEMBL29206981 0.72 KMT2A (0.44) KMT2AMAPTNPC1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2164833-B1 Quinazolinamide derivatives useful for the treatment of tumour diseases MERCK PATENT GMBH (DE) 2015-04-15 EP disclosed