SCHEMBL16650004

SCHEMBL16650004

NC(=O)OCCOC[CH]c1ccc(F)c(Cl)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.35
IDO1 P14902 1/20 0.35
LMNA P02545 1/20 0.33
TSHR P16473 1/20 0.33
CASP1 P29466 1/20 0.33
PYGL P06737 1/20 0.33
DPEP1 P16444 1/20 0.32
ICMT O60725 1/20 0.32
SLC2A1 P11166 1/20 0.32
HDAC3 O15379 1/20 0.32
HDAC4 P56524 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC7 Q8WUI4 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC10 Q969S8 1/20 0.32
HDAC11 Q96DB2 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
HDAC9 Q9UKV0 1/20 0.32
HDAC5 Q9UQL6 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16649545 0.88 TRPA1 (0.39) TRPA1IDO1TSHRCASP1DPEP1
SCHEMBL16649875 0.82 ALDH1A1 (0.39) TRPA1IDO1TSHRCASP1DPEP1
SCHEMBL16649314 0.80 IDO1 (0.36) TRPA1IDO1LMNATSHRPYGL
SCHEMBL12498864 0.76 KCNA3 (0.37)
SCHEMBL15157522 0.74 TRPA1 (0.41) TRPA1IDO1TSHRCASP1DPEP1
SCHEMBL16649568 0.74 ALDH1A1 (0.48) LMNAPYGLMAPTKMT2A
SCHEMBL16649643 0.74 ALDH1A1 (0.48) PYGLMAPTKMT2A
SCHEMBL16649920 0.74 TSHR (0.39) TRPA1IDO1LMNATSHRDPEP1
SCHEMBL12498442 0.71 IDO1 (0.41) TRPA1IDO1LMNATSHRPYGL
SCHEMBL16961107 0.70 TRPA1 (0.43) TRPA1TSHRHDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9133187-B2 Serine/threonine kinase inhibitors ARRAY BIOPHARMA INC. (US) 2015-09-15 US claimed
EP-2681215-B1 SERINE/THREONINE KINASE INHIBITORS ARRAY BIOPHARMA INC (US) 2015-04-22 EP claimed