SCHEMBL1665019

SCHEMBL1665019

O=C(Cn1ccc2cc(NC(=O)c3ccc(-n4ccc5cc(Nc6ccc(N7CCC(O)CC7)cc6)ccc54)cc3)ccc21)NC1CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNIK Q9UKE5 1/20 0.41
ALDH1A1 P00352 4/20 0.39
KDM4E B2RXH2 3/20 0.39
HPGD P15428 2/20 0.39
LMNA P02545 2/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
KRAS P01116 4/20 0.38
NPY5R Q15761 4/20 0.38
SMYD3 Q9H7B4 2/20 0.37
EPHX2 P34913 1/20 0.36
DHODH Q02127 1/20 0.36
TSHR P16473 2/20 0.35
HSD17B10 Q99714 2/20 0.35
USP2 O75604 2/20 0.35
POLB P06746 2/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1665021 0.97 ALDH1A1 (0.41) TNIKALDH1A1KDM4EHPGDLMNA
SCHEMBL1665971 0.88 JAK2 (0.41) TNIKALDH1A1HPGDNPSR1RXFP1
SCHEMBL1664054 0.87 TNIK (0.42) TNIKALDH1A1KDM4ELMNAEPHX2
SCHEMBL1666783 0.86 SMYD3 (0.46) TNIKSMYD3DHODHMAPTSYK
SCHEMBL1666784 0.86 SMYD3 (0.46) TNIKKDM4ELMNASMYD3EPHX2
SCHEMBL8775930 0.85 PIN1 (0.42) TNIKALDH1A1LMNAEPHX2DHODH
SCHEMBL1665973 0.84 MEN1 (0.40) TNIKALDH1A1HPGDNPSR1RXFP1
SCHEMBL1666719 0.83 MAPT (0.39) TNIKALDH1A1KDM4EHPGDLMNA
SCHEMBL1664050 0.83 DHODH (0.42) TNIKALDH1A1LMNAEPHX2DHODH
SCHEMBL1664697 0.82 MAPT (0.41) TNIKALDH1A1KDM4EHPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2488486-A1 HEMATOPOIETIC GROWTH FACTOR MIMETIC SMALL MOLECULE COMPOUNDS AND THEIR USES Ligand Pharmaceuticals Inc. (US) 2012-08-22 EP disclosed
WO-2011046954-A1 HEMATOPOIETIC GROWTH FACTOR MIMETIC SMALL MOLECULE COMPOUNDS AND THEIR USES LIGAND PHARMACEUTICALS INC. (US) 2011-04-21 WO disclosed