SCHEMBL16655975

SCHEMBL16655975

CS(=O)(=O)Oc1ccccc1-c1cnco1

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 17/20 0.44
IMPDH1 P20839 2/20 0.44
AAK1 Q2M2I8 2/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
POLB P06746 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1906120 0.79 IMPDH2 (0.62) IMPDH2IMPDH1AAK1
SCHEMBL16655599 0.77 NOTUM (0.36) IMPDH2IMPDH1POLBKMT2A
SCHEMBL29664573 0.77 NOTUM (0.36) IMPDH2IMPDH1POLBKMT2A
SCHEMBL29866188 0.76 NPC1 (0.42) POLBKMT2A
SCHEMBL29866032 0.75 NPC1 (0.41) POLBKMT2A
SCHEMBL343458 0.70 EDNRB (0.43) IMPDH2IMPDH1CYP11B1CYP11B2POLB
SCHEMBL10767560 0.70 ALOX5AP (0.43) IMPDH2IMPDH1CYP11B1CYP11B2POLB
SCHEMBL3839152 0.70 NFE2L2 (0.42) KMT2A
SCHEMBL10035045 0.70 IMPDH2 (0.51) IMPDH2IMPDH1AAK1CYP11B1CYP11B2
SCHEMBL1363022 0.70 NOTUM (0.50) IMPDH2IMPDH1CYP11B1CYP11B2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3383183-A1 MIXTURES OF CIS-JASMONE ANDBACILLUS AMYLOLIQUEFACIENS BASF SE (DE) 2018-10-10 EP claimed
EP-3206490-A1 METHOD AND PESTICIDAL MIXTURES FOR CONTROLLING PENTATOMIDAE PESTS BASF SE (DE) 2017-08-23 EP claimed
WO-2017093163-A1 MIXTURES OF CIS-JASMONE AND BACILLUS AMYLOLIQUEFACIENS BASF SE (DE) 2017-06-08 WO claimed
WO-2016059240-A1 METHOD AND PESTICIDAL MIXTURES FOR CONTROLLING PENTATOMIDAE PESTS BASF SE (DE) 2016-04-21 WO claimed
EP-3534709-A1 SUBSTITUTED SULFONYL AMIDES FOR CONTROLLING ANIMAL PESTS Bayer Aktiengesellschaft (DE) 2019-09-11 EP disclosed
EP-3523299-A1 2-(HET)ARYL-SUBSTITUTED CONDENSED BICYCLIC HETEROCYCLE DERIVATIVES AS PEST CONTROL AGENTS Bayer CropScience Aktiengesellschaft (DE) 2019-08-14 EP disclosed
EP-3515921-A1 PYRAZOLO [1,5-A]PYRIDINE DERIVATIVES AND THEIR USE AS PESTICIDES Bayer CropScience Aktiengesellschaft (DE) 2019-07-31 EP disclosed
EP-3497102-A1 CONDENSED BICYCLIC HETEROCYCLE DERIVATIVES AS PEST CONTROL AGENTS Bayer CropScience Aktiengesellschaft (DE) 2019-06-19 EP disclosed
EP-3487860-A1 CONDENSED BICYCLIC HETEROCYCLE DERIVATIVES AS PEST CONTROL AGENTS Bayer CropScience Aktiengesellschaft (DE) 2019-05-29 EP disclosed
EP-3426044-A1 FUNGICIDAL MIXTURES III COMPRISING STROBILURIN-TYPE FUNGICIDES BASF SE (DE) 2019-01-16 EP disclosed
EP-3419418-A1 SOLVENT-FREE FORMULATIONS OF LOW-MELTING ACTIVE SUBSTANCES Bayer CropScience Aktiengesellschaft (DE) 2019-01-02 EP disclosed
EP-3414237-A1 SUBSTITUTED 2-OXYIMIDAZOLYL-CARBOXAMIDES AS PEST CONTROL AGENTS Bayer CropScience Aktiengesellschaft (DE) 2018-12-19 EP disclosed
EP-3402797-A1 HETEROCYCLENE DERIVATIVES AS PEST CONTROL AGENTS Bayer CropScience AG (DE) 2018-11-21 EP disclosed
EP-3383874-A1 MESOIONIC HALOGENATED 3-(ACETYL)-1-[(1,3-THIAZOL-5-YL)METHYL]-1H-IMIDAZO[1,2-A]PYRIDIN-4-IUM-2-OLATE DERIVATIVES AND RELATED COMPOUNDS AS INSECTICIDES Bayer CropScience Aktiengesellschaft (DE) 2018-10-10 EP disclosed
WO-2017153200-A1 FUNGICIDAL MIXTURES III COMPRISING STROBILURIN-TYPE FUNGICIDES BASF SE (DE) 2017-09-14 WO disclosed
EP-3206490-A1 METHOD AND PESTICIDAL MIXTURES FOR CONTROLLING PENTATOMIDAE PESTS BASF SE (DE) 2017-08-23 EP disclosed
EP-3057424-A1 ACTIVE COMPOUND COMBINATIONS COMPRISING A (THIO)CARBOXAMIDE DERIVATIVE AND A FUNGICIDAL COMPOUND Bayer CropScience Aktiengesellschaft (DE) 2016-08-24 EP disclosed
WO-2016059240-A1 METHOD AND PESTICIDAL MIXTURES FOR CONTROLLING PENTATOMIDAE PESTS BASF SE (DE) 2016-04-21 WO disclosed
WO-2015055707-A9 ACTIVE COMPOUND COMBINATIONS COMPRISING A (THIO)CARBOXAMIDE DERIVATIVE AND A FUNGICIDAL COMPOUND BAYER CROPSCIENCE AG (DE) 2015-07-02 WO disclosed
WO-2015055707-A1 ACTIVE COMPOUND COMBINATIONS COMPRISING A (THIO)CARBOXAMIDE DERIVATIVE AND A FUNGICIDAL COMPOUND BAYER CROPSCIENCE AG (DE) 2015-04-23 WO disclosed