SCHEMBL16656117

SCHEMBL16656117

Cc1ncc(C(=O)c2ccc3nc(Cl)c(-c4ccccc4)c(Cl)c3c2)[nH]1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
RORC P51449 18/20 0.43
ALDH1A1 P00352 1/20 0.40
POLB P06746 1/20 0.40
HPGD P15428 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
FABP3 P05413 1/20 0.38
FABP4 P15090 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16632084 0.78 RORC (0.56) RORC
SCHEMBL15647202 0.75 RORC (0.55) RORCALDH1A1FABP3FABP4
SCHEMBL15647176 0.75 RORC (0.48) RORCALDH1A1RAB9ASMN1; SMN2FABP3
SCHEMBL16633049 0.74 RORC (0.56) RORC
SCHEMBL16655904 0.71 RORC (0.66) RORC
SCHEMBL15201636 0.70 TAS1R3 (0.40) ALDH1A1RAB9ASMN1; SMN2
SCHEMBL15646319 0.70 NAPRT (0.50) ALDH1A1POLBRAB9ASMN1; SMN2
SCHEMBL22726319 0.69 RORC (0.56) RORC
SCHEMBL16653816 0.69 RAB9A (0.46) HPGDRAB9ASMN1; SMN2
SCHEMBL18754799 0.69 RORC (0.45) RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057421-A1 ALKYL LINKED QUINOLINYL MODULATORS OF ROR(GAMMA)T Janssen Pharmaceutica, N.V. (BE) 2016-08-24 EP disclosed
WO-2015057629-A1 ALKYL LINKED QUINOLINYL MODULATORS OF RORyt JANSSEN PHARMACEUTICA NV (BE) 2015-04-23 WO disclosed