SCHEMBL16660906

SCHEMBL16660906

CC=C(CBr)c1c(F)cccc1C(F)(F)F

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
STIM1 Q13586 1/20 0.34
ORAI1 Q96D31 1/20 0.34
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
ITGA4 P13612 3/20 0.33
RORC P51449 3/20 0.33
ITGB1 P05556 2/20 0.33
PTGS2 P35354 1/20 0.33
HSD11B1 P28845 1/20 0.33
RORB Q92753 1/20 0.32
TRPA1 O75762 2/20 0.32
CTSS P25774 1/20 0.32
TDP1 Q9NUW8 2/20 0.32
P2RX7 Q99572 1/20 0.32
CYP1A2 P05177 1/20 0.32
CNR2 P34972 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2096065 0.77 CES2 (0.44) STIM1ORAI1CES2CES1ITGA4
SCHEMBL20428863 0.73 STIM1 (0.36) STIM1ORAI1CES2CES1ITGA4
SCHEMBL716995 0.70 CES2 (0.48) STIM1ORAI1CES2CES1RORC
SCHEMBL30313345 0.70 CES2 (0.48) STIM1ORAI1CES2CES1RORC
SCHEMBL14534757 0.70 CES2 (0.39) STIM1ORAI1CES2CES1ITGA4
SCHEMBL4710152 0.70 CES2 (0.44) STIM1ORAI1CES2CES1ITGA4
SCHEMBL5358162 0.68 PTPN1 (0.48) CTSSCNR2
SCHEMBL7939207 0.68 RORC (0.42) STIM1ORAI1CES2CES1ITGA4
SCHEMBL503596 0.68 CES2 (0.50) STIM1ORAI1CES2CES1ITGA4
SCHEMBL20560651 0.67 CES2 (0.39) STIM1ORAI1CES2CES1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2862856-A1 AROMATIC HETEROCYCLIC COMPOUND Mitsubishi Tanabe Pharma Corporation (JP) 2015-04-22 EP disclosed