SCHEMBL1666355

SCHEMBL1666355

FC(F)(F)c1nc2ccccc2s1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASR P41180 10/20 0.50
PIK3CG P48736 1/20 0.49
PSMB8 P28062 1/20 0.48
PSMB5 P28074 1/20 0.48
ALDH1A1 P00352 1/20 0.48
ADRA2A P08913 1/20 0.48
FBP1 P09467 1/20 0.48
ADORA3 P0DMS8 1/20 0.48
DRD2 P14416 1/20 0.48
HPGD P15428 1/20 0.48
ALOX15 P16050 1/20 0.48
ADRA2B P18089 1/20 0.48
ADRA2C P18825 1/20 0.48
DRD1 P21728 1/20 0.48
MC5R P33032 1/20 0.48
OPRM1 P35372 1/20 0.48
DRD3 P35462 1/20 0.48
OPRK1 P41145 1/20 0.48
CCR2 P41597 1/20 0.48
HTR6 P50406 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7738337 0.84 CASR (0.47) CASRPIK3CGPSMB8PSMB5ALDH1A1
SCHEMBL28366070 0.81 CASR (0.45) CASRPIK3CGPSMB8PSMB5ALDH1A1
SCHEMBL5720317 0.81 CASR (0.51) CASRPSMB8PSMB5ALDH1A1ADRA2A
SCHEMBL28370247 0.80 CASR (0.44) CASRPIK3CGPSMB8PSMB5ALDH1A1
SCHEMBL227210 0.79 CASR (0.58) CASRALDH1A1ADRA2AFBP1ADORA3
SCHEMBL3907554 0.79 CASR (0.53) CASRPSMB8PSMB5ALDH1A1ADRA2A
SCHEMBL108180 0.79 CASR (0.58) CASRALDH1A1ADRA2AFBP1ADORA3
SCHEMBL28366681 0.78 CASR (0.43) CASRPIK3CGPSMB8PSMB5ALDH1A1
SCHEMBL7544923 0.76 CASR (0.64) CASRALDH1A1ADRA2AFBP1ADORA3
SCHEMBL6120718 0.75 MIF (0.49) ALDH1A1ALOX15HSD17B10TDP1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 78 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119552155-A Trifluoromethyl benzothiazole tertiary alcohol derivative and preparation method and application thereof 河南农业大学 2025-03-04 CN claimed
US-10224485-B2 Process for preparing a crystalline organic semiconductor material BASF SE (DE) 2019-03-05 US claimed
US-4939140-A ALDOSE REDUCTASE INHIBITORS PFIZER INC. (US) 1990-07-03 US claimed
US-20260132119-A1 Alkylphenyl Substituted Compounds, Compositions and Methods of Use DEEP APPLE THERAPEUTICS, INC. (US) 2026-05-14 US disclosed
CN-119552155-B Trifluoromethyl benzothiazole tertiary alcohol derivative and preparation method and application thereof 河南农业大学 2025-11-04 CN disclosed
CN-119552155-B Trifluoromethyl benzothiazole tertiary alcohol derivative and preparation method and application thereof 河南农业大学 2025-11-04 CN disclosed
CN-119552155-A Trifluoromethyl benzothiazole tertiary alcohol derivative and preparation method and application thereof 河南农业大学 2025-03-04 CN disclosed
CN-119552155-A Trifluoromethyl benzothiazole tertiary alcohol derivative and preparation method and application thereof 河南农业大学 2025-03-04 CN disclosed
CN-119552155-A Trifluoromethyl benzothiazole tertiary alcohol derivative and preparation method and application thereof 河南农业大学 2025-03-04 CN disclosed
US-20250066344-A1 BENZOTHIAZOLE, BENZOISOXAZOLE, AND BENZODIOXOLE ANALOGS AS RXFP1 RECEPTOR AGONISTS BRISTOL MYERS SQUIBB CO (US) 2025-02-27 US disclosed
EP-4448500-A1 BENZOTHIAZOLE, BENZOISOXAZOLE AND BENZODIOXOLE ANALOGS AS RXFP1 RECEPTOR AGONISTS Bristol-Myers Squibb Company (US) 2024-10-23 EP disclosed
US-7141596-B2 Inhibitors of proteins that bind phosphorylated molecules INCYTE CORPORATION (US) 2006-11-28 US disclosed
CN-1760190-A Method for preparing trifluoromethyl benzothiazole UNIV SHANGHAI (CN) 2006-04-19 CN disclosed
CN-1760190-A Method for preparing trifluoromethyl benzothiazole UNIV SHANGHAI (CN) 2006-04-19 CN disclosed
US-20050272778-A1 Inhibitors of proteins that bind phosphorylated molecules INCYTE CORPORATION 2005-12-08 US disclosed
EP-0565579-B1 2-IMINO 6-POLYFLUORALKYL 3-HETEROCYCLYLALKYL BENZOTHIAZOLINE DERIVATIVES, THEIR PREPARATION AND DRUGS CONTAINING SAME RHONE POULENC RORER SA (FR) 1994-07-20 EP disclosed
EP-0565579-A1 2-IMINO 6-POLYFLUORALKYL 3-HETEROCYCLYLALKYL BENZOTHIAZOLINE DERIVATIVES, THEIR PREPARATION AND DRUGS CONTAINING SAME. RHONE POULENC RORER SA (FR) 1993-10-20 EP disclosed
EP-0374040-B1 2-IMINO-BENZOTHIAZOLINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM RHONE-POULENC SANTE (FR) 1993-03-24 EP disclosed
WO-1992012142-A1 2-IMINO 6-POLYFLUORALKYL 3-HETEROCYCLYLALKYL BENZOTHIAZOLINE DERIVATIVES, THEIR PREPARATION AND DRUGS CONTAINING SAME RHONE-POULENC RORER S.A. (FR) 1992-07-23 WO disclosed
EP-0374040-A1 2-Imino-benzothiazoline derivatives, processes for their preparation and medicaments containing them RHONE-POULENC SANTE (FR) 1990-06-20 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050272778-A1 Inhibitors of proteins that bind phosphorylated molecules PPP3CA, PPP5C, PPM1A CASR 3633/4885PIK3CG 341/4885PSMB8 1288/4885
US-20260132119-A1 Alkylphenyl Substituted Compounds, Compositions and Methods of Use GIPR, MC2R, GRPR CASR 623/4885PIK3CG 1838/4885PSMB8 2182/4885
US-10224485-B2 Process for preparing a crystalline organic semiconductor material STOM, SPOP, TTR CASR 880/4885PIK3CG 1204/4885PSMB8 4668/4885
US-20250066344-A1 BENZOTHIAZOLE, BENZOISOXAZOLE, AND BENZODIOXOLE ANALOGS AS RXFP1 RECEPTOR AGONISTS RXFP1, RXFP2, RXFP3 CASR 963/4885PIK3CG 4335/4885PSMB8 2830/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.