SCHEMBL16665019

SCHEMBL16665019

CCNc1cc(-c2ccc(NC3CCN(CC(F)(F)F)CC3)nc2)ncn1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 1/20 0.44
HPGDS O60760 7/20 0.43
TBK1 Q9UHD2 4/20 0.41
SYK P43405 5/20 0.40
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
IKBKE Q14164 1/20 0.39
CCNK O75909 1/20 0.38
CDK12 Q9NYV4 1/20 0.38
CCR6 P51684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19819913 0.92 HPGDS (0.44) TDO2HPGDSTBK1SYKCNR1
SCHEMBL15473152 0.89 FLT3 (0.42) HPGDSTBK1CNR1CNR2
SCHEMBL15473174 0.86 TDO2 (0.46) TDO2TBK1SYKCCNKCDK12
SCHEMBL16664942 0.86 SYK (0.49) TDO2TBK1SYKIKBKECCNK
SCHEMBL15343201 0.84 PIK3CA (0.41) TDO2TBK1SYKCCR6
SCHEMBL16664992 0.83 CDK1 (0.41) HPGDSTBK1SYKIKBKE
SCHEMBL15473175 0.82 HPGDS (0.43) HPGDSTBK1IKBKE
SCHEMBL16664999 0.80 HPGDS (0.36) HPGDSTBK1IKBKE
SCHEMBL19819895 0.79 TDO2 (0.44) TDO2TBK1SYKCCNKCDK12
SCHEMBL15473156 0.76 CDK1 (0.40) HPGDSTBK1SYKIKBKE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015058031-A1 DNA-PK INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2015-04-23 WO disclosed