SCHEMBL16664942

SCHEMBL16664942

CCNc1cc(-c2ccc(NC3CCN(C)CC3)nc2)ncn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 4/20 0.49
TBK1 Q9UHD2 2/20 0.44
HRH4 Q9H3N8 1/20 0.43
DYRK1A Q13627 5/20 0.43
GSK3B P49841 3/20 0.43
TDO2 P48775 1/20 0.41
PIK3CA P42336 2/20 0.41
FLT3 P36888 1/20 0.40
TYRO3 Q06418 1/20 0.40
MERTK Q12866 1/20 0.40
GAS6 Q14393 1/20 0.40
CLK2 P49760 1/20 0.40
CLK3 P49761 1/20 0.40
CCNT1 O60563 1/20 0.40
CCNK O75909 2/20 0.39
CDK12 Q9NYV4 2/20 0.39
IKBKE Q14164 1/20 0.39
NOS3 P29474 1/20 0.39
NOS1 P29475 1/20 0.39
NOS2 P35228 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15343201 0.89 PIK3CA (0.41) SYKTBK1DYRK1AGSK3BTDO2
SCHEMBL15473155 0.86 FLT3 (0.46) SYKTBK1HRH4FLT3TYRO3
SCHEMBL16665019 0.86 TDO2 (0.44) SYKTBK1TDO2CCNKCDK12
SCHEMBL15473174 0.86 TDO2 (0.46) SYKTBK1DYRK1AGSK3BTDO2
SCHEMBL15473069 0.81 TBK1 (0.40) SYKTBK1HRH4DYRK1AGSK3B
SCHEMBL19355355 0.81 CYP1A2 (0.47) SYKHRH4GSK3BFLT3TYRO3
SCHEMBL15356477 0.80 KIT (0.50) PIK3CA
SCHEMBL15356381 0.80 ALDH1A1 (0.41) SYKTBK1DYRK1AGSK3BPIK3CA
SCHEMBL20373137 0.80 CYP3A4 (0.42) SYKDYRK1AGSK3BFLT3TYRO3
SCHEMBL17634517 0.80 CYP3A4 (0.42) SYKDYRK1AGSK3BFLT3TYRO3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015058031-A1 DNA-PK INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2015-04-23 WO disclosed