SCHEMBL16670549

SCHEMBL16670549

COc1ccc(N(Cc2ccccc2)C(=O)C(Cc2ccccc2)NC(=O)O)cc1

nearest known ligand 0.62

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTPRB P23467 1/20 0.57
RNF4 P78317 1/20 0.54
TRPM8 Q7Z2W7 1/20 0.53
FPR2 P25090 1/20 0.51
KMT2A Q03164 2/20 0.49
ALDH1A1 P00352 1/20 0.49
LMNA P02545 1/20 0.49
MEN1 O00255 1/20 0.49
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
ACHE P22303 1/20 0.47
PYGL P06737 1/20 0.46
PPARG P37231 1/20 0.46
PPARA Q07869 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20427718 0.87 PTPRB (0.56) PTPRBRNF4TRPM8FPR2PPARG
SCHEMBL16682060 0.87 PTPRB (0.56) PTPRBRNF4TRPM8FPR2PPARG
SCHEMBL16670186 0.85 FPR2 (0.53) FPR2KMT2AALDH1A1NPC1RAB9A
SCHEMBL16670359 0.83 PTPRB (0.51) PTPRBRNF4TRPM8FPR2KMT2A
SCHEMBL16670358 0.83 PTPRB (0.51) PTPRBRNF4TRPM8FPR2KMT2A
SCHEMBL16682042 0.81 RNF4 (0.57) RNF4TRPM8KMT2AALDH1A1LMNA
SCHEMBL16669947 0.81 RNF4 (0.57) RNF4TRPM8KMT2AALDH1A1LMNA
SCHEMBL16682162 0.81 FPR2 (0.54) PTPRBTRPM8FPR2KMT2AALDH1A1
SCHEMBL16670145 0.79 PTPRB (0.47) PTPRBRNF4TRPM8FPR2KMT2A
SCHEMBL16670144 0.79 PTPRB (0.47) PTPRBRNF4TRPM8FPR2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10035760-B2 Inhibitors of human immunodeficiency virus replication VIIV HEALTHCARE UK (NO. 5) LIMITED (GB) 2018-07-31 US disclosed
US-20160257645-A1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION VIIV Healthcare UK (No.5) Limited (GB) 2016-09-08 US disclosed
EP-3060554-A1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION Bristol-Myers Squibb Company (US) 2016-08-31 EP disclosed
WO-2015061518-A1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION BRISTOL-MYERS SQUIBB COMPANY (US) 2015-04-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160257645-A1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION EIF2AK2, POLR1E, POLR1G PTPRB 3674/4885RNF4 1646/4885TRPM8 4660/4885
US-10035760-B2 Inhibitors of human immunodeficiency virus replication EIF2AK2, POLR1G, POLR1E PTPRB 3692/4885RNF4 1773/4885TRPM8 4685/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.