SCHEMBL16684

SCHEMBL16684

NCCCC[C@H](N)C(=O)OC(=O)OC(=O)[C@@H](N)CCCCN

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GSR P00390 1/20 0.57
GNAI3 P08754 1/20 0.41
GNAO1 P09471 1/20 0.41
GNAI1 P63096 1/20 0.41
RNPEP Q9H4A4 1/20 0.41
DPP7 Q9UHL4 8/20 0.40
DPP8 Q6V1X1 4/20 0.40
DPP9 Q86TI2 4/20 0.40
DPP4 P27487 2/20 0.40
CPB2 Q96IY4 4/20 0.40
FAP Q12884 1/20 0.36
CYP1A2 P05177 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27655247 0.98 GSR (0.55) GSRGNAI3GNAO1GNAI1RNPEP
SCHEMBL28456987 0.98 GSR (0.55) GSRGNAI3GNAO1GNAI1RNPEP
SCHEMBL28091506 0.94 GSR (0.48) GSRGNAI3GNAO1GNAI1RNPEP
SCHEMBL344574 0.91 GSR (0.61) GSRGNAI3GNAO1GNAI1RNPEP
SCHEMBL20240364 0.91 GSR (0.61) GSRGNAI3GNAO1GNAI1RNPEP
SCHEMBL1404247 0.91 GSR (0.61) GSRGNAI3GNAO1GNAI1RNPEP
SCHEMBL680614 0.89 GSR (0.59) GSRGNAI3GNAO1GNAI1RNPEP
Hydrochloric Acid SCHEMBL2099474 0.89 GSR (0.59) GSRGNAI3GNAO1GNAI1RNPEP
Hydrochloric Acid SCHEMBL3825519 0.89 GSR (0.59) GSRGNAI3GNAO1GNAI1RNPEP
SCHEMBL16194521 0.89 GSR (0.59) GSRGNAI3GNAO1GNAI1RNPEP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2535 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250332107-A1 IMMEDIATE RELEASE DOSAGE FORM KENVUE BRANDS LLC (US) 2025-10-30 US claimed
CN-120058564-A Method and device for producing pentanediol 摩珈(上海)生物科技有限公司 2025-05-30 CN claimed
US-12296049-B2 Immediate release dosage form KENVUE BRANDS LLC (US) 2025-05-13 US claimed
CN-106714783-B Effervescent composition and method for preparing same 驶帝生命科学印度私人有限公司 2025-04-18 CN claimed
WO-2025040153-A1 METHOD FOR PREPARING ISOCYANATE AND DEVICE 摩珈(上海)生物科技有限公司 2025-02-27 WO claimed
EP-4473962-A2 IMMEDIATE RELEASE DOSAGE FORM Johnson & Johnson Consumer Inc. (US) 2024-12-11 EP claimed
EP-3781136-B1 IMMEDIATE RELEASE DOSAGE FORM JOHNSON & JOHNSON CONSUMER INC (US) 2024-09-25 EP claimed
US-20240180821-A1 ORALLY DISINTEGRATING FILM COMPOSITION OF KETOROLAC AND A METHOD OF PREPARATION THEREOF LN LABORATORIES PVT LTD (IN) 2024-06-06 US claimed
US-20230414520-A1 IMMEDIATE RELEASE DOSAGE FORM KENVUE BRANDS LLC 2023-12-28 US claimed
US-20230293633-A1 Apoaequorin and Curcumin Containing Compositions and Methods QUINCY BIOSCIENCE, LLC 2023-09-21 US claimed
US-6319683-B1 CARBONYLATION WITH FORMALDEHYDE INTERGEN COMPANY 2001-11-20 US claimed
US-6248361-B1 MIXTURE OF FOLIC ACID WITH CARBONATE INTEG, LTD. 2001-06-19 US claimed
WO-2001022917-A2 EFFERVESCENT COMPOSITIONS COMPRISING NIMESULIDE PANACEA BIOTEC LIMITED (IN) 2001-04-05 WO claimed
US-6072086-A QUENCHING AQUEOUS FORMALDEHYDE SOLUTION WITH COMPOSITION COMPRISING FIRST AGENT CAPABLE OF REACTING WITH FORMALDEHYDE, SECOND AGENT CAPABLE OF SUBSTANTIALLY PREVENTING FIRST AGENT FROM REACTING WITH FORMALDEHYDE FOR FINITE TIME PERIOD INTERGEN COMPANY (US) 2000-06-06 US claimed
EP-0954292-A1 PHARMACEUTICAL FORMULATIONS WITH DELAYED DRUG RELEASE POLI INDUSTRIA CHIMICA S.p.A. (IT) 1999-11-10 EP claimed
US-5788987-A TIME-SPECIFIC CONTROLLED RELEASE DOSAGE FORMULATION POLI INDUSTRIA CHIMICA SPA (IT) 1998-08-04 US claimed
WO-1998032425-A1 PHARMACEUTICAL FORMULATIONS WITH DELAYED DRUG RELEASE POLI INDUSTRIA CHIMICA S.P.A. (US) 1998-07-30 WO claimed
EP-0155427-B1 READY FOR USE, RAPIDLY DISINTEGRATING, SOLID CULTURE MEDIUM, AND PROCESS FOR ITS PREPARATION SOCIETE D'APPLICATIONS PHARMACEUTIQUES ET BIOLOGIQUES HOECHST-BEHRING (FR) 1988-05-04 EP claimed
EP-0092287-B1 ACETYLCYSTEINE SALTS, THEIR PREPARATION AND USE "PHARLYSE", Société Anonyme (LU) 1987-03-25 EP claimed
EP-0078785-B1 SALTS OF VALPROIC ACID, THEIR PREPARATION AND THEIR USE "PHARLYSE", Société Anonyme (LU) 1985-04-03 EP claimed