SCHEMBL16684159

SCHEMBL16684159

CN(C)CCOc1cc2cc(S(=O)(=O)NCP(=O)(O)Oc3ccc(C#N)c(C(F)(F)F)c3)sc2cc1OCCN

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PLA2G7 Q13093 2/20 0.33
AR P10275 8/20 0.33
UTS2R Q9UKP6 1/20 0.32
SLC22A12 Q96S37 1/20 0.32
TRPV4 Q9HBA0 1/20 0.31
KDR P35968 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13031987 0.94 SLC22A12 (0.34) PLA2G7ARSLC22A12TRPV4
Trifluoroacetic Acid SCHEMBL3948690 0.91 PLA2G7 (0.34) PLA2G7ARSLC22A12TRPV4
SCHEMBL14943082 0.91 SLC22A12 (0.34) PLA2G7ARSLC22A12TRPV4
Trifluoroacetic Acid SCHEMBL4158728 0.87 CACNA1B (0.36) PLA2G7ARSLC22A12
SCHEMBL13032081 0.86 TRPV4 (0.36) PLA2G7ARSLC22A12TRPV4
SCHEMBL13031985 0.85 TRPV4 (0.36) TRPV4
SCHEMBL16684145 0.84 AR (0.33) PLA2G7ARTRPV4
SCHEMBL16684158 0.83 CYP1A2 (0.32) AR
SCHEMBL14942995 0.83 CYP1A2 (0.32) AR
SCHEMBL14943083 0.81 TRPV4 (0.36) TRPV4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049200-B1 NOVEL INHIBITORS OF BETA-LACTAMASE METHYLGENE INC (CA) 2015-04-29 EP disclosed