SCHEMBL16684604

SCHEMBL16684604

O=Cc1ccc2occ(C(F)(F)F)c2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.42
KIF11 P52732 2/20 0.41
PTPN1 P18031 8/20 0.40
PTPN2 P17706 1/20 0.34
KDM4E B2RXH2 3/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
AKR1C3 P42330 1/20 0.33
AKR1C2 P52895 1/20 0.33
ERN1 O75460 1/20 0.33
ALDH1A1 P00352 3/20 0.33
HSD17B10 Q99714 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
PTGS2 P35354 1/20 0.32
RAB9A P51151 1/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16686997 0.80 ALDH1A1 (0.40) KDM4EMEN1KMT2AALDH1A1CA12
SCHEMBL16686996 0.80 ALDH1A1 (0.40) KDM4EMEN1KMT2AALDH1A1CA12
SCHEMBL16684571 0.77 PTPN1 (0.46) CYP2A6KIF11PTPN1PTPN2KDM4E
SCHEMBL17345173 0.74 KIF11 (0.53) CYP2A6KIF11KDM4EMEN1KMT2A
SCHEMBL23241583 0.74 TP53 (0.46) KIF11MAOAMAOBALDH1A1CA12
SCHEMBL2883176 0.74 ALDH1A1 (0.46) CYP2A6PTPN1PTPN2KDM4EMEN1
SCHEMBL1852687 0.74 PTPN1 (0.46) CYP2A6KIF11PTPN1PTPN2KDM4E
SCHEMBL16684629 0.74 PTPN1 (0.46) PTPN1MEN1KMT2AMAOAMAOB
SCHEMBL472408 0.70 KIF11 (0.56) CYP2A6KIF11KDM4EAKR1C3AKR1C2
SCHEMBL18235043 0.70 PTPN1 (0.47) CYP2A6PTPN1PTPN2KDM4EMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015066371-A1 SPIRO-OXADIAZOLINE COMPOUNDS AS AGONISTS OF α-7-NICOTINIC ACETYLCHOLINE RECEPTORS FORUM PHARMACEUTICALS, INC. (US) 2015-05-07 WO disclosed
WO-2015066371-A1 SPIRO-OXADIAZOLINE COMPOUNDS AS AGONISTS OF α-7-NICOTINIC ACETYLCHOLINE RECEPTORS FORUM PHARMACEUTICALS, INC. (US) 2015-05-07 WO disclosed