SCHEMBL16701338

SCHEMBL16701338

Nc1nc(N)c(C2CC2)c(-c2ccc(C(F)(F)F)cc2)n1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HEXA P06865 1/20 0.46
HEXB P07686 1/20 0.46
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
DPP4 P27487 1/20 0.40
KIF11 P52732 2/20 0.40
PLAU P00749 1/20 0.39
HRH4 Q9H3N8 1/20 0.39
KCNH2 Q12809 5/20 0.38
DHFR P00374 2/20 0.37
MYC P01106 1/20 0.37
WDR5 P61964 1/20 0.37
PDE8B O95263 1/20 0.37
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
MEN1 O00255 1/20 0.36
MAPT P10636 1/20 0.36
BLM P54132 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16701358 0.93 HEXA (0.43) HEXAHEXBMKNK1MKNK2DPP4
SCHEMBL28152107 0.83 ADORA2A (0.53) DHFRADORA2AADORA1MEN1KMT2A
SCHEMBL28151073 0.79 ADORA2A (0.51) ADORA2AADORA1MEN1KMT2A
SCHEMBL12137851 0.79 ADORA2A (0.51) ADORA2AADORA1MEN1MAPTKMT2A
SCHEMBL28151079 0.77 ADORA1 (0.52) HEXAHEXBDHFRADORA2AADORA1
SCHEMBL27631813 0.76 HEXA (0.51) HEXAHEXBMKNK1MKNK2DPP4
SCHEMBL27942788 0.75 HEXA (0.54) HEXAHEXBMKNK1MKNK2DPP4
SCHEMBL16703371 0.75 RAF1 (0.45) ADORA2AADORA1
SCHEMBL28152086 0.73 DHFR (0.47) DHFRADORA2AADORA1
SCHEMBL10456198 0.72 MTOR (0.65) HEXAHEXBMKNK1MKNK2DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015069752-A9 ACETYLCHOLINE BINDING PROTEIN LIGANDS, COOPERATIVE NACHR MODULATORS AND METHODS FOR MAKING AND USING THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2015-07-09 WO disclosed
WO-2015069752-A1 ACETYLCHOLINE BINDING PROTEIN LIGANDS, COOPERATIVE NACHR MODULATORS AND METHODS FOR MAKING AND USING THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2015-05-14 WO disclosed