SCHEMBL16701358

SCHEMBL16701358

Nc1nc(N)c(C2CCCCCC2)c(-c2ccc(C(F)(F)F)cc2)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HEXA P06865 1/20 0.43
HEXB P07686 1/20 0.43
MKNK1 Q9BUB5 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38
PLAU P00749 2/20 0.38
DPP4 P27487 1/20 0.38
TNK2 Q07912 1/20 0.37
GABBR2 O75899 3/20 0.37
GABBR1 Q9UBS5 3/20 0.37
KIF11 P52732 1/20 0.37
MAPK13 O15264 1/20 0.36
RAF1 P04049 1/20 0.36
MAPK9 P45984 1/20 0.36
MAPK12 P53778 1/20 0.36
MAPK11 Q15759 1/20 0.36
MAPK14 Q16539 1/20 0.36
HRH4 Q9H3N8 1/20 0.36
RPS6KB1 P23443 1/20 0.36
AKT1 P31749 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16701338 0.93 HEXA (0.46) HEXAHEXBMKNK1MKNK2PLAU
SCHEMBL12137851 0.83 ADORA2A (0.51) TNK2MAPK13MAPK9MAPK12MAPK11
SCHEMBL16703371 0.83 RAF1 (0.45) MAPK13RAF1MAPK9MAPK12MAPK11
SCHEMBL28152086 0.81 DHFR (0.47) TNK2DHFR
SCHEMBL28151073 0.81 ADORA2A (0.51) TNK2MAPK13MAPK9MAPK12MAPK11
SCHEMBL28152107 0.77 ADORA2A (0.53) MAPK13MAPK9MAPK12MAPK11MAPK14
SCHEMBL28152025 0.77 HRH3 (0.53) HEXAHEXBTNK2DHFR
SCHEMBL28267193 0.74 HRH3 (0.53) HEXAHEXBTNK2DHFR
SCHEMBL27631813 0.73 HEXA (0.51) HEXAHEXBMKNK1MKNK2PLAU
SCHEMBL27942788 0.72 HEXA (0.54) HEXAHEXBMKNK1MKNK2PLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015069752-A9 ACETYLCHOLINE BINDING PROTEIN LIGANDS, COOPERATIVE NACHR MODULATORS AND METHODS FOR MAKING AND USING THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2015-07-09 WO disclosed
WO-2015069752-A1 ACETYLCHOLINE BINDING PROTEIN LIGANDS, COOPERATIVE NACHR MODULATORS AND METHODS FOR MAKING AND USING THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2015-05-14 WO disclosed