SCHEMBL16705126

SCHEMBL16705126

N#Cc1ccc(Nc2ccc(Br)cc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.57
MAOA P21397 1/20 0.57
IDO1 P14902 3/20 0.56
LMNA P02545 1/20 0.50
MAPT P10636 1/20 0.50
MEN1 O00255 1/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
KMT2A Q03164 1/20 0.45
CA2 P00918 2/20 0.44
CA1 P00915 1/20 0.44
CYP1B1 Q16678 1/20 0.42
ABCG2 Q9UNQ0 4/20 0.42
ABCB1 P08183 3/20 0.42
DHODH Q02127 1/20 0.42
MMP2 P08253 1/20 0.41
SYK P43405 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP2A6 P11509 1/20 0.41
CA12 O43570 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL395539 0.88 CA2 (0.52) IDO1LMNAMAPTMEN1RAB9A
SCHEMBL154636 0.85
Water SCHEMBL27994834 0.85 MAOB (0.73) MAOBMAOAIDO1CA2CA1
SCHEMBL6827721 0.83 MAOB (0.70) MAOBMAOAIDO1CA2CA1
Hydrochloric Acid SCHEMBL30722972 0.83 MAOB (0.70) MAOBMAOAIDO1CA2CA1
SCHEMBL14656590 0.83 MAOB (0.70) MAOBMAOAIDO1CA2CA1
SCHEMBL25546850 0.81 MMP3 (0.56) CA2CA1CYP1B1ABCG2ABCB1
SCHEMBL16526973 0.80 CYP2A6 (0.57) MAOBMAOAIDO1LMNAMAPT
SCHEMBL13148721 0.80 CYP2A6 (0.57) MAOBMAOAIDO1LMNAMAPT
SCHEMBL409605 0.80 CYP2A6 (0.57) MAOBMAOAIDO1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9029353-B2 Boron-containing small molecules as anti-inflammatory agents ANACOR PHARMACEUTICALS, INC. (US) 2015-05-12 US disclosed