SCHEMBL16705198

SCHEMBL16705198

COc1ccc(C2(c3ccc(O)cc3)C=Cc3c4c(c5cc(OC)ccc5c3O2)-c2ccc(-c3cncnc3)cc2C4(C)C)cc1

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 3/20 0.34
CYP11B1 P15538 3/20 0.34
CYP11B2 P19099 3/20 0.34
BACE1 P56817 10/20 0.34
KCNH2 Q12809 4/20 0.34
KMT2A Q03164 1/20 0.34
CYP3A4 P08684 2/20 0.33
PDE4D Q08499 1/20 0.32
CTSD P07339 2/20 0.32
NCOA1 Q15788 1/20 0.31
NCOA3 Q9Y6Q9 1/20 0.31
FYN P06241 2/20 0.31
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15028836 0.96 CYP17A1 (0.37) CYP17A1CYP11B1CYP11B2BACE1KCNH2
SCHEMBL15028784 0.90 ESR1 (0.36) BACE1KMT2APDE4D
SCHEMBL9926882 0.90 ESR1 (0.37) BACE1KMT2APDE4D
SCHEMBL9897952 0.89 BACE1 (0.33) CYP17A1CYP11B1CYP11B2BACE1KCNH2
SCHEMBL9928451 0.89 BACE1 (0.33) CYP17A1CYP11B1CYP11B2BACE1KCNH2
SCHEMBL9899115 0.86 KDM4E (0.34) BACE1KMT2ACYP3A4
SCHEMBL16705204 0.85 ESR1 (0.36) BACE1KMT2APDE4D
SCHEMBL25607194 0.83 KDM4E (0.33) BACE1KMT2A
SCHEMBL16705200 0.82 PDK2 (0.31) PDE4D
SCHEMBL25844764 0.82 ALKBH3 (0.33) BACE1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9028728-B2 Photochromic materials that include indeno-fused naphthopyrans TRANSITIONS OPTICAL, INC. (US) 2015-05-12 US disclosed