SCHEMBL16705221

SCHEMBL16705221

CCOC(=O)c1nc(CC)sc1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.47
CYP1A2 P05177 2/20 0.47
GAA P10253 2/20 0.42
MAPT P10636 3/20 0.41
NPC1 O15118 1/20 0.41
TP53 P04637 1/20 0.41
XBP1 P17861 1/20 0.41
MAPK1 P28482 1/20 0.41
HTT P42858 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TLR9 Q9NR96 1/20 0.41
GLP1R P43220 1/20 0.40
TARBP2 Q15633 1/20 0.40
TRPM8 Q7Z2W7 1/20 0.40
HPGD P15428 3/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
LMNA P02545 2/20 0.39
KDM4E B2RXH2 1/20 0.39
GABRA2 P47869 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12849586 0.87 ALDH1A1 (0.45) ALDH1A1CYP1A2GAAMAPTNPC1
SCHEMBL18792316 0.87 ALDH1A1 (0.45) ALDH1A1CYP1A2GAAMAPTNPC1
SCHEMBL10350633 0.87 ALDH1A1 (0.45) ALDH1A1CYP1A2GAAMAPTNPC1
SCHEMBL18792315 0.84 ALDH1A1 (0.43) ALDH1A1CYP1A2GAAMAPTNPC1
SCHEMBL27832378 0.83 KMT2A (0.33) ALDH1A1CYP1A2GAANPC1MAPK1
SCHEMBL28397631 0.83 MEN1 (0.42) ALDH1A1CYP1A2GAAMAPTNPC1
SCHEMBL9861374 0.83 ALDH1A1 (0.50) ALDH1A1CYP1A2GAAMAPTNPC1
SCHEMBL6505364 0.83 GAA (0.55) ALDH1A1CYP1A2GAAMAPTNPC1
SCHEMBL10317272 0.83 ALDH1A1 (0.50) ALDH1A1CYP1A2GAAMAPTNPC1
SCHEMBL595444 0.81 ALDH1A1 (0.49) ALDH1A1CYP1A2GAAMAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2620433-B1 SUBSTITUTED AMIDE COMPOUND ASTELLAS PHARMA INC (JP) 2015-05-13 EP disclosed