SCHEMBL16709409

SCHEMBL16709409

Cc1ccc(-n2c(-c3nonc3N)noc2=O)cc1Br

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.42
RPS6KB1 P23443 7/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
ROCK1 Q13464 2/20 0.36
GSK3B P49841 4/20 0.36
PRKACA P17612 2/20 0.36
RPS6KA5 O75582 5/20 0.35
ALDH1A1 P00352 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
LMNA P02545 1/20 0.34
GAA P10253 1/20 0.34
HTT P42858 1/20 0.33
ALKBH5 Q6P6C2 1/20 0.33
THRB P10828 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29030690 0.87 IDO1 (0.42) IDO1RPS6KB1ROCK1GSK3BPRKACA
SCHEMBL123581 0.87 IDO1 (0.54) IDO1RPS6KB1ROCK1GSK3BPRKACA
SCHEMBL29376679 0.87 IDO1 (0.54) IDO1RPS6KB1ROCK1GSK3BPRKACA
SCHEMBL29030673 0.86 RPS6KB1 (0.43) IDO1RPS6KB1L3MBTL1ROCK1GSK3B
SCHEMBL19661056 0.85 PKM (0.39) IDO1RPS6KB1L3MBTL1ROCK1GSK3B
SCHEMBL29030697 0.84 RPS6KB1 (0.38) IDO1RPS6KB1ROCK1GSK3BPRKACA
SCHEMBL16706551 0.83 IDO1 (0.42) IDO1RPS6KB1ROCK1GSK3BPRKACA
SCHEMBL21326485 0.82 IDO1 (0.44) IDO1RPS6KB1ROCK1GSK3BPRKACA
SCHEMBL22001225 0.82 IDO1 (0.38) IDO1RPS6KB1ROCK1GSK3BPRKACA
SCHEMBL21118338 0.80 PTGS1 (0.37) IDO1RPS6KB1ROCK1GSK3BPRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110343098-B Oxadiazole compound, preparation method, pharmaceutical composition and application thereof 中国科学院上海药物研究所 2023-05-26 CN disclosed
WO-2015070007-A1 PROCESS FOR THE SYNTHESIS OF AN INDOLEAMINE 2,3-DIOXYGENASE INHIBITOR INCYTE CORPORATION (US) 2015-05-14 WO disclosed