SCHEMBL29030673

SCHEMBL29030673

COc1ccc(-n2c(-c3nonc3N)noc2=O)cc1Br

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RPS6KB1 P23443 5/20 0.43
ROCK1 Q13464 4/20 0.43
IDO1 P14902 1/20 0.40
BRD9 Q9H8M2 2/20 0.38
CYP2C9 P11712 1/20 0.38
TSHR P16473 2/20 0.36
HCRTR1 O43613 1/20 0.36
HCRTR2 O43614 1/20 0.36
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
KMT2A Q03164 4/20 0.36
LMNA P02545 1/20 0.36
RPS6KA5 O75582 1/20 0.36
PRKACA P17612 2/20 0.36
GSK3B P49841 2/20 0.36
ALDH1A1 P00352 2/20 0.36
HPGD P15428 1/20 0.36
AMY1A P0DUB6 1/20 0.36
MEN1 O00255 3/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16709409 0.86 IDO1 (0.42) RPS6KB1ROCK1IDO1HTTLMNA
SCHEMBL123581 0.83 IDO1 (0.54) RPS6KB1ROCK1IDO1NPSR1KMT2A
SCHEMBL29030690 0.83 IDO1 (0.42) RPS6KB1ROCK1IDO1CYP2C9TSHR
SCHEMBL29376679 0.83 IDO1 (0.54) RPS6KB1ROCK1IDO1NPSR1KMT2A
SCHEMBL29030746 0.81 RPS6KB1 (0.62) RPS6KB1ROCK1TSHRKMT2ALMNA
SCHEMBL21326485 0.78 IDO1 (0.44) RPS6KB1ROCK1IDO1NPSR1KMT2A
SCHEMBL22001225 0.78 IDO1 (0.38) RPS6KB1ROCK1IDO1HTTRPS6KA5
SCHEMBL29030697 0.78 RPS6KB1 (0.38) RPS6KB1ROCK1IDO1KMT2ARPS6KA5
SCHEMBL29043089 0.77 RPS6KB1 (0.42) RPS6KB1ROCK1IDO1CYP2C9TSHR
SCHEMBL19661056 0.77 PKM (0.39) RPS6KB1ROCK1IDO1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110343098-B Oxadiazole compound, preparation method, pharmaceutical composition and application thereof 中国科学院上海药物研究所 2023-05-26 CN disclosed